SCHEMBL10685115

SCHEMBL10685115

[CH2]C1CCCN(CC2CC2)C1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 1/20 0.46
ADRA2C P18825 1/20 0.46
KDM2B Q8NHM5 15/20 0.40
SCN1A P35498 1/20 0.39
SCN4A P35499 1/20 0.39
SCN7A Q01118 1/20 0.39
KCNH2 Q12809 1/20 0.39
SCN5A Q14524 1/20 0.39
SCN9A Q15858 1/20 0.39
SCN2A Q99250 1/20 0.39
SCN3A Q9NY46 1/20 0.39
SCN11A Q9UI33 1/20 0.39
SCN8A Q9UQD0 1/20 0.39
SCN10A Q9Y5Y9 1/20 0.39
DRD2 P14416 1/20 0.39
DRD3 P35462 1/20 0.39
ACHE P22303 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1202306 0.92 CHRM5 (0.59) CHRM5ADRA2CKDM2BACHE
SCHEMBL1202459 0.92 CHRM5 (0.59) CHRM5ADRA2CKDM2BACHE
SCHEMBL1201943 0.92 CHRM5 (0.59) CHRM5ADRA2CKDM2BACHE
SCHEMBL478537 0.86 CHRM5 (0.39) CHRM5ADRA2CSCN1ASCN4ASCN7A
SCHEMBL772390 0.76
SCHEMBL3667628 0.75 KCNH2 (0.40) CHRM5ADRA2CKDM2BKCNH2DRD3
SCHEMBL12717548 0.74 ACHE (0.50) CHRM5ADRA2CKDM2BSCN1ASCN4A
SCHEMBL19807339 0.74 CHRM5 (0.46) CHRM5ADRA2CKDM2BSCN1ASCN4A
SCHEMBL21120886 0.74 ALDH1A1 (0.49) CHRM5ADRA2CKDM2BSCN1ASCN4A
SCHEMBL21120881 0.74 ACHE (0.50) CHRM5ADRA2CKDM2BSCN1ASCN4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4780478-A Aminopropoxy-chromones useful as antidepressants MERCK PATENT GESELLSCHAFT MIT BERSCHRANKTER HAFTUNG (DE) 1988-10-25 US disclosed
US-4508732-A Basic ethers useful as antidepressant agents MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1985-04-02 US disclosed
EP-0031885-B1 BASIC ETHERS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESS FOR THEIR PREPARATION MERCK PATENT GmbH (DE) 1984-06-27 EP disclosed
US-4376123-A Hexahydroazepinyloxy-chromones useful as antidepressants MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1983-03-08 US disclosed
EP-0031885-A1 Basic ethers, pharmaceutical compositions containing them and process for their preparation MERCK PATENT GmbH (DE) 1981-07-15 EP disclosed