SCHEMBL10686138

SCHEMBL10686138

CC(C)(C)C(=O)C(C#N)c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.45
AKR1C3 P42330 1/20 0.45
AKR1C1 Q04828 1/20 0.45
TSHR P16473 1/20 0.44
CTSS P25774 2/20 0.41
CTSK P43235 1/20 0.41
HSP90AA1 P07900 1/20 0.41
MAPT P10636 1/20 0.41
GPR55 Q9Y2T6 1/20 0.41
CNR1 P21554 1/20 0.41
CNR2 P34972 1/20 0.41
CYP3A4 P08684 1/20 0.40
HIF1A Q16665 1/20 0.40
TRPA1 O75762 1/20 0.39
CTSL P07711 1/20 0.39
CTSB P07858 1/20 0.39
POLB P06746 2/20 0.39
HTT P42858 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
KDM4E B2RXH2 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10686874 0.82 BRD4 (0.41) ALDH1A1TSHRMAPTCNR1CYP3A4
SCHEMBL6097343 0.81 TSHR (0.44) ALDH1A1AKR1C3AKR1C1TSHRCTSS
SCHEMBL8764471 0.79 TSHR (0.41) ALDH1A1AKR1C3AKR1C1TSHRCTSS
SCHEMBL1720075 0.79 ALDH1A1 (0.49) ALDH1A1AKR1C3AKR1C1TSHRCYP3A4
SCHEMBL11813692 0.78 TSHR (0.52) ALDH1A1AKR1C3AKR1C1TSHRTRPA1
SCHEMBL1019171 0.78 TSHR (0.52) ALDH1A1AKR1C3AKR1C1TSHRTRPA1
SCHEMBL409758 0.78 POLB (0.50) ALDH1A1HSP90AA1MAPTGPR55CYP3A4
SCHEMBL15268630 0.77 CTSS (0.48) ALDH1A1AKR1C3AKR1C1TSHRCTSS
SCHEMBL6960576 0.76 TSHR (0.50) ALDH1A1AKR1C3AKR1C1TSHRTRPA1
Ammonia Solution, Strong SCHEMBL38661532 0.76 TSHR (0.50) ALDH1A1AKR1C3AKR1C1TSHRTRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4716237-A Process for the production of 3-oxonitriles DEGUSSA AKTIENGESELLSCHAFT (DE) 1987-12-29 US claimed
US-4728743-A Process for the production of 3-oxonitriles DEGUSSA AKTIENGESELLSCHAFT (DE) 1988-03-01 US disclosed
US-4716237-A Process for the production of 3-oxonitriles DEGUSSA AKTIENGESELLSCHAFT (DE) 1987-12-29 US disclosed
EP-0089011-B1 PROCESS FOR THE PREPARATION OF 5-OXONITRILES Degussa Aktiengesellschaft (DE) 1985-07-10 EP disclosed
EP-0089011-A1 Process for the preparation of 5-oxonitriles Degussa Aktiengesellschaft (DE) 1983-09-21 EP disclosed