SCHEMBL10690101

SCHEMBL10690101

COc1ccccc1C1Cc2ccccc2NC1=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.48
TSHR P16473 3/20 0.48
TDP1 Q9NUW8 3/20 0.48
LMNA P02545 1/20 0.48
HPGD P15428 1/20 0.48
PKM P14618 1/20 0.48
BRD4 O60885 1/20 0.44
CREBBP Q92793 1/20 0.44
MEN1 O00255 4/20 0.43
KMT2A Q03164 4/20 0.43
USP2 O75604 1/20 0.43
POLB P06746 1/20 0.43
CYP19A1 P11511 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
MAPT P10636 2/20 0.42
RECQL P46063 2/20 0.42
TP53 P04637 1/20 0.42
GAA P10253 1/20 0.42
HSD17B10 Q99714 1/20 0.42
MAPK1 P28482 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6275913 0.78 BRD4 (0.44) ALDH1A1TSHRLMNAHPGDBRD4
SCHEMBL6280031 0.77 DDB1 (0.54) ALDH1A1LMNAHPGDPKMBRD4
SCHEMBL7286888 0.77 ALDH1A1 (0.43) ALDH1A1TSHRTDP1LMNAHPGD
SCHEMBL2003982 0.74 DDB1 (0.59) ALDH1A1LMNABRD4CREBBPMEN1
SCHEMBL25575861 0.74 DDB1 (0.66) ALDH1A1TSHRTDP1LMNAHPGD
SCHEMBL5668502 0.73 DDB1 (0.50) ALDH1A1TSHRTDP1HPGDBRD4
SCHEMBL6252884 0.72 BRD4 (0.47) ALDH1A1TDP1LMNAHPGDBRD4
SCHEMBL10691415 0.70 DRD2 (0.44) ALDH1A1TDP1PKMMEN1KMT2A
SCHEMBL5783641 0.70 CREBBP (0.49) ALDH1A1TSHRBRD4CREBBPMEN1
SCHEMBL6221253 0.70 CREBBP (0.61) TSHRBRD4CREBBPMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4778793-A CONTROLLING CALCIUM CONCENTRATION-CARDIOVASCULAR DISORDERS HOECHST AKTIENGESELLSCHAFT (DE) 1988-10-18 US disclosed
EP-0212216-A1 Dihydroquinolinone derivatives, processes for their preparation, medicaments containing them, the use of these medicaments, and intermediates for their preparation HOECHST AKTIENGESELLSCHAFT (DE) 1987-03-04 EP disclosed