SCHEMBL10691415

SCHEMBL10691415

COc1ccccc1C1Cc2ccccc2N(C)C1=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.44
DRD3 P35462 2/20 0.44
HTR2C P28335 4/20 0.43
ADRA2A P08913 1/20 0.43
ADRA2B P18089 1/20 0.43
ADRA2C P18825 1/20 0.43
SLC6A2 P23975 1/20 0.43
HTR2A P28223 1/20 0.43
SLC6A4 P31645 1/20 0.43
ADRA1A P35348 1/20 0.43
HRH1 P35367 1/20 0.43
HTR2B P41595 1/20 0.43
KCNH2 Q12809 1/20 0.43
ALDH1A1 P00352 3/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
KDM4E B2RXH2 1/20 0.43
USP2 O75604 1/20 0.43
POLB P06746 1/20 0.43
GAA P10253 1/20 0.43
THRB P10828 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10694704 0.80 DRD2 (0.40) DRD2DRD3HTR2CADRA2AADRA2B
SCHEMBL10688450 0.80 ADRA1A (0.46) DRD2HTR2CADRA2AADRA2BADRA2C
SCHEMBL10694512 0.78 CACNA1S (0.51) CYP19A1MEN1KMT2A
Hydrochloric Acid SCHEMBL10690626 0.77 HTR1A (0.45) DRD2HTR2AADRA1AALDH1A1KDM4E
SCHEMBL30489285 0.76 TSHR (0.65) DRD2HTR2CADRA2AADRA2BADRA2C
SCHEMBL10695532 0.76 TSHR (0.65) DRD2HTR2CADRA2AADRA2BADRA2C
SCHEMBL10368739 0.75 HSD11B1 (0.45) ALDH1A1L3MBTL1KDM4EUSP2GAA
SCHEMBL10691585 0.75 LMNA (0.49) ALDH1A1KDM4EGAAHSD17B10CYP19A1
SCHEMBL13495369 0.72 CYP19A1 (0.45) ALDH1A1L3MBTL1USP2RECQLCYP19A1
SCHEMBL9560256 0.71 MAPT (0.56) DRD2HTR2CADRA2AADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4778793-A CONTROLLING CALCIUM CONCENTRATION-CARDIOVASCULAR DISORDERS HOECHST AKTIENGESELLSCHAFT (DE) 1988-10-18 US disclosed
EP-0212216-A1 Dihydroquinolinone derivatives, processes for their preparation, medicaments containing them, the use of these medicaments, and intermediates for their preparation HOECHST AKTIENGESELLSCHAFT (DE) 1987-03-04 EP disclosed