SCHEMBL10690347

SCHEMBL10690347

Nc1nc(N)c2c(N)cccc2n1

nearest known ligand 0.66

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
DCPS Q96C86 3/20 0.59
DHFR P00374 10/20 0.54
KCNH2 Q12809 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1154870 0.81 DCPS (0.58) DCPSDHFRKCNH2
SCHEMBL3340224 0.79 DCPS (0.61) DCPSDHFRKCNH2
SCHEMBL29224081 0.79 DCPS (0.56) DCPSDHFRKCNH2
SCHEMBL30912748 0.79 DHFR (0.57) DCPSDHFRKCNH2
SCHEMBL8390061 0.79 DHFR (0.66) DCPSDHFRKCNH2
SCHEMBL29740318 0.79 DCPS (0.61) DCPSDHFRKCNH2
SCHEMBL2127622 0.79 DHFR (0.57) DCPSDHFRKCNH2
SCHEMBL30912751 0.79 DHFR (0.66) DCPSDHFRKCNH2
SCHEMBL8222792 0.76 DCPS (0.72) DCPSDHFRKCNH2
SCHEMBL30482707 0.75 DHFR (0.58) DCPSDHFRKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-86100512-A 2 of antitumor action is arranged, and 4-diamino-6-(N-methyl or formyl radical-replacement benzyl amino) quinoline derivatives is synthetic 1987-09-02 CN claimed
WO-2016201219-A1 SMALL MOLECULE INHIBITORS OF DIHYDROFOLATE REDUCTASE CIDARA THERAPEUTICS, INC. (US) 2016-12-15 WO disclosed
US-20160117440-A1 SYSTEM AND METHOD FOR AUTOMATED PREDICTION OF VULNERABILITIES IN BIOLOGICAL SAMPLES MEMORIAL SLOAN-KETTERING CANCER CENTER 2016-04-28 US disclosed
CN-1049498-A 2,4-diamino-5-replacement-6-(N-replaces benzyl amino) quinazoline derivant is synthetic SHANGHAI INST PHARM INDUSTRY (CN) 1991-02-27 CN disclosed
CN-1049498-A 2,4-diamino-5-replacement-6-(N-replaces benzyl amino) quinazoline derivant is synthetic SHANGHAI INST PHARM INDUSTRY (CN) 1991-02-27 CN disclosed
EP-0253396-A2 Process for preparing 5,6-substituted-2,4-quinazolinediamines and intermediates WARNER-LAMBERT COMPANY (US) 1988-01-20 EP disclosed