SCHEMBL10691711

SCHEMBL10691711

[c]1c(Cc2cccnc2)ccc2ccccc12

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 2/20 0.41
CYP11B2 P19099 2/20 0.41
HRH4 Q9H3N8 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
CYP2D6 P10635 4/20 0.40
CYP1A2 P05177 2/20 0.40
CYP3A4 P08684 2/20 0.39
SLC6A2 P23975 2/20 0.39
SLC6A4 P31645 2/20 0.39
SLC6A3 Q01959 2/20 0.39
KCNH2 Q12809 2/20 0.39
MMP2 P08253 1/20 0.39
CHRNA7 P36544 1/20 0.39
TBXAS1 P24557 2/20 0.38
LTA4H P09960 1/20 0.38
IDO1 P14902 1/20 0.38
CHRNB2 P17787 2/20 0.38
CHRNA4 P43681 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL852825 0.81 CALM1 (0.42) CYP2D6CYP1A2LTA4H
SCHEMBL11863358 0.77 CYP2A6 (0.32) CYP1A2
SCHEMBL11014831 0.71 L3MBTL1 (0.40) HRH4HRH3
SCHEMBL727185 0.71 CYP1A2 (0.62) CYP11B1CYP11B2HRH4HRH3CYP2D6
SCHEMBL3959322 0.70 CYP11B1 (0.45) CYP11B1CYP11B2HRH4HRH3CYP2D6
SCHEMBL28233327 0.70 CYP11B1 (0.53) CYP11B1CYP11B2HRH4HRH3CYP2D6
SCHEMBL29995759 0.69 CYP11B1 (0.65) CYP11B1CYP11B2HRH4HRH3CYP2D6
SCHEMBL177863 0.69 CYP11B1 (0.65) CYP11B1CYP11B2HRH4HRH3CYP2D6
SCHEMBL6740961 0.69 KCNH2 (0.39) KCNH2
SCHEMBL6704132 0.69 CYP11B1 (0.50) CYP11B1CYP11B2CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4734406-A 3-pyridylmethylnaphthyl derivatives and composition containing them useful to inhibit thromboxane synthetase HOECHST AKTIENGESELLSCHAFT (DE) 1988-03-29 US disclosed
EP-0194579-A2 3-Pyridylmethylnaphthyl derivatives, process for their preparation and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1986-09-17 EP disclosed