SCHEMBL10692018

SCHEMBL10692018

CCN(Cc1cnc2nc(N)nc(N)c2c1C)c1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 9/20 0.62
KDM4E B2RXH2 1/20 0.62
TLR4 O00206 1/20 0.62
MEN1 O00255 1/20 0.62
ALDH1A1 P00352 1/20 0.62
LMNA P02545 1/20 0.62
TP53 P04637 1/20 0.62
TYMS P04818 1/20 0.62
GLA P06280 1/20 0.62
POLB P06746 1/20 0.62
HMGB1 P09429 1/20 0.62
MAPT P10636 1/20 0.62
FOLR2 P14207 1/20 0.62
FOLR1 P15328 1/20 0.62
HPGD P15428 1/20 0.62
ALOX15 P16050 1/20 0.62
ALOX12 P18054 1/20 0.62
GART P22102 1/20 0.62
APEX1 P27695 1/20 0.62
CASP1 P29466 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1073086 0.85 DHFR (0.83) DHFRKDM4ETLR4MEN1ALDH1A1
SCHEMBL2794954 0.85 DHFR (0.83) DHFRKDM4ETLR4MEN1ALDH1A1
SCHEMBL9765067 0.83 DHFR (0.71) DHFRTYMSFOLR1SLC19A1SLC46A1
SCHEMBL8325555 0.79 DHFR (0.54) DHFRKDM4ETLR4MEN1ALDH1A1
SCHEMBL10697242 0.78 DHFR (0.63) DHFRKDM4ETLR4MEN1ALDH1A1
SCHEMBL10691004 0.77 DHFR (0.56) DHFRKDM4ETLR4MEN1ALDH1A1
SCHEMBL5321065 0.77 DHFR (0.71) DHFRKDM4ETLR4MEN1ALDH1A1
Methotrexate SCHEMBL171251 0.77 DHFR (1.00) DHFRKDM4ETLR4MEN1ALDH1A1
Methotrexate SCHEMBL3712 0.77 DHFR (1.00) DHFRKDM4ETLR4MEN1ALDH1A1
Methotrexate SCHEMBL20548444 0.77 DHFR (1.00) DHFRKDM4ETLR4MEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4725687-A ANTITUMOR AGENTS; SIDE EFFECT REDUCTION; POTENCY SOUTHERN RESEARCH INSTITUTE (US) 1988-02-16 US disclosed