SCHEMBL8325555

SCHEMBL8325555

Cc1c(CN(C)c2ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)s2)cnc2nc(N)nc(N)c12

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 4/20 0.54
TYMS P04818 2/20 0.54
FOLR2 P14207 2/20 0.54
FOLR1 P15328 2/20 0.54
SLC19A1 P41440 2/20 0.54
SLC46A1 Q96NT5 2/20 0.54
NCOA3 Q9Y6Q9 2/20 0.54
KDM4E B2RXH2 1/20 0.54
TLR4 O00206 1/20 0.54
MEN1 O00255 1/20 0.54
ALDH1A1 P00352 1/20 0.54
LMNA P02545 1/20 0.54
TP53 P04637 1/20 0.54
GLA P06280 1/20 0.54
POLB P06746 1/20 0.54
HMGB1 P09429 1/20 0.54
MAPT P10636 1/20 0.54
HPGD P15428 1/20 0.54
ALOX15 P16050 1/20 0.54
ALOX12 P18054 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9067195 0.91 DHFR (0.51) DHFRTYMSFOLR2FOLR1SLC19A1
SCHEMBL8326393 0.84 TYMS (0.51) DHFRTYMSGART
SCHEMBL10692018 0.79 DHFR (0.62) DHFRTYMSFOLR2FOLR1SLC19A1
SCHEMBL31143667 0.78 DHFR (0.62) DHFRTYMSFOLR2FOLR1SLC19A1
SCHEMBL9041174 0.76 DHFR (0.55) DHFRTYMSFOLR2FOLR1SLC19A1
SCHEMBL9844872 0.76 TYMS (0.52) DHFRTYMSFOLR2FOLR1SLC19A1
SCHEMBL9765067 0.75 DHFR (0.71) DHFRTYMSFOLR1SLC19A1SLC46A1
SCHEMBL8325682 0.75 GART (0.49) DHFRTYMSGART
SCHEMBL9227335 0.75 TYMS (0.51) DHFRTYMSFOLR2FOLR1SLC19A1
SCHEMBL10691004 0.73 DHFR (0.56) DHFRTYMSFOLR2FOLR1SLC19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0638079-B1 DEAZAAMINOPTERINS FOR TREATMENT OF INFLAMMATION STANFORD RES INST INT (US) 1999-12-15 EP disclosed
US-5536724-A Antiinflammatory and antineoplastic 5-deazaaminopterins and 5,10-dideazaaminopterins SRI INTERNATIONAL (US) 1996-07-16 US disclosed