SCHEMBL10693130

SCHEMBL10693130

COc1ccccc1C1(O)C(=O)N(C)c2ccccc2C1O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.43
TSHR P16473 2/20 0.43
SCN9A Q15858 1/20 0.42
HSD11B1 P28845 6/20 0.41
HTT P42858 2/20 0.40
KMT2A Q03164 2/20 0.40
MAPT P10636 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
MAPK1 P28482 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
GPR55 Q9Y2T6 1/20 0.39
RAD52 P43351 1/20 0.39
CHRM2 P08172 1/20 0.38
CHRM4 P08173 1/20 0.38
CHRM5 P08912 1/20 0.38
CHRM1 P11229 1/20 0.38
CHRM3 P20309 1/20 0.38
TP53 P04637 1/20 0.37
PKM P14618 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL841729 0.71 MAPT (0.44) ALDH1A1TSHRHSD11B1HTTKMT2A
SCHEMBL10370674 0.68 RAD52 (0.48) ALDH1A1TSHRSCN9AHTTKMT2A
SCHEMBL31389171 0.67 TSHR (0.58) ALDH1A1TSHRHTTKMT2AMAPT
SCHEMBL10368739 0.66 HSD11B1 (0.45) ALDH1A1HSD11B1KMT2AMAPTKDM4E
SCHEMBL27524948 0.66 SCN9A (0.62) ALDH1A1SCN9AKMT2ATP53
SCHEMBL10689170 0.66 ADRA1A (0.40) ALDH1A1TSHRSCN9AHSD11B1HTT
SCHEMBL29475767 0.65 PDK2 (0.42) ALDH1A1HSD11B1KMT2AMAPTKDM4E
SCHEMBL10370026 0.65 SCN9A (0.43) ALDH1A1TSHRSCN9AHSD11B1HTT
SCHEMBL10691597 0.63 ADRA1A (0.39) ALDH1A1TSHRSCN9AMAPTRAD52
SCHEMBL10690604 0.63 TDP1 (0.42) ALDH1A1TSHRSCN9AMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4778793-A CONTROLLING CALCIUM CONCENTRATION-CARDIOVASCULAR DISORDERS HOECHST AKTIENGESELLSCHAFT (DE) 1988-10-18 US disclosed
EP-0212216-A1 Dihydroquinolinone derivatives, processes for their preparation, medicaments containing them, the use of these medicaments, and intermediates for their preparation HOECHST AKTIENGESELLSCHAFT (DE) 1987-03-04 EP disclosed