SCHEMBL10691597

SCHEMBL10691597

COc1ccccc1C1(C(C)C)Cc2ccccc2N(C)C1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 4/20 0.39
ADRA1D P25100 3/20 0.39
ADRA1B P35368 3/20 0.39
RAD52 P43351 1/20 0.38
ALDH1A1 P00352 3/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
DRD2 P14416 1/20 0.38
DRD3 P35462 1/20 0.38
GAA P10253 1/20 0.37
CASP3 P42574 1/20 0.37
CASP6 P55212 1/20 0.37
SENP8 Q96LD8 1/20 0.37
SENP7 Q9BQF6 1/20 0.37
SENP6 Q9GZR1 1/20 0.37
SCN9A Q15858 1/20 0.37
TSHR P16473 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
ADRA2B P18089 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10694665 0.83 RAD52 (0.36) ADRA1AADRA1DADRA1BRAD52ALDH1A1
SCHEMBL10693548 0.82 RAD52 (0.35) ADRA1AADRA1DADRA1BRAD52ALDH1A1
SCHEMBL10695401 0.82 RAD52 (0.42) RAD52ALDH1A1MAPTTSHRADAMTS5
SCHEMBL10691306 0.81 ALDH1A1 (0.41) RAD52ALDH1A1MAPTTSHRTDP1
SCHEMBL10696619 0.81 RAD52 (0.34) ADRA1AADRA1DADRA1BRAD52ALDH1A1
SCHEMBL10689170 0.81 ADRA1A (0.40) ADRA1AADRA1DADRA1BALDH1A1MAPT
SCHEMBL10691593 0.80 L3MBTL1 (0.42) ALDH1A1MAPTSCN9ATSHRL3MBTL1
SCHEMBL10690604 0.78 TDP1 (0.42) ADRA1AADRA1DADRA1BALDH1A1MAPT
Hydrochloric Acid SCHEMBL10758557 0.77 DRD2 (0.41) ADRA1AADRA1DADRA1BALDH1A1DRD2
Hydrochloric Acid SCHEMBL10695756 0.75 MEN1 (0.47) ALDH1A1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4778793-A CONTROLLING CALCIUM CONCENTRATION-CARDIOVASCULAR DISORDERS HOECHST AKTIENGESELLSCHAFT (DE) 1988-10-18 US disclosed
EP-0212216-A1 Dihydroquinolinone derivatives, processes for their preparation, medicaments containing them, the use of these medicaments, and intermediates for their preparation HOECHST AKTIENGESELLSCHAFT (DE) 1987-03-04 EP disclosed