SCHEMBL10693536

SCHEMBL10693536

CC(=O)Cn1cnc2c1c(=O)n(CCC(C)O)c(=O)n2CCC(C)O

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 6/20 0.71
PDE4B Q07343 5/20 0.71
PDE4C Q08493 5/20 0.71
PDE4D Q08499 5/20 0.71
ADORA2B P29275 4/20 0.71
ADORA2A P29274 2/20 0.71
TRPA1 O75762 3/20 0.59
SMN1; SMN2 Q16637 3/20 0.49
LMNA P02545 2/20 0.49
ALDH1A1 P00352 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
ESR1 P03372 1/20 0.47
CYP1A2 P05177 1/20 0.47
MAPT P10636 1/20 0.47
NFKB1 P19838 1/20 0.47
ACHE P22303 1/20 0.47
BLM P54132 1/20 0.47
PMP22 Q01453 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10694979 0.93 PDE4A (0.84) PDE4APDE4BPDE4CPDE4DADORA2B
SCHEMBL10694974 0.93 PDE4A (0.84) PDE4APDE4BPDE4CPDE4DADORA2B
SCHEMBL9682937 0.86 TRPA1 (0.65) PDE4APDE4BPDE4CPDE4DADORA2B
SCHEMBL10696123 0.85 PDE4A (0.76) PDE4APDE4BPDE4CPDE4DADORA2B
SCHEMBL10694067 0.85 SMN1; SMN2 (0.67) PDE4APDE4BPDE4CPDE4DADORA2B
Denbufylline SCHEMBL127152 0.83 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DADORA2B
Denbufylline SCHEMBL7299526 0.83 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DADORA2B
Denbufylline SCHEMBL11044404 0.82 PDE4A (0.97) PDE4APDE4BPDE4CPDE4DADORA2B
SCHEMBL10872056 0.81 PDE4A (0.95) PDE4APDE4BPDE4CPDE4DADORA2B
SCHEMBL7323464 0.80 PDE4A (0.93) PDE4APDE4BPDE4CPDE4DADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0260127-A2 Xanthine derivatives, their preparation and pharmaceutical compositions containing them BEECHAM - WUELFING GmbH & Co. KG (DE) 1988-03-16 EP claimed
EP-0260127-A2 Xanthine derivatives, their preparation and pharmaceutical compositions containing them BEECHAM - WUELFING GmbH & Co. KG (DE) 1988-03-16 EP disclosed