SCHEMBL9682937

SCHEMBL9682937

CC(=O)Cn1cnc2c1c(=O)n(CCCCC(C)O)c(=O)n2C

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 5/20 0.65
PDE4A P27815 4/20 0.63
ADORA2B P29275 4/20 0.63
PDE4B Q07343 3/20 0.63
PDE4C Q08493 3/20 0.63
PDE4D Q08499 3/20 0.63
ADORA2A P29274 1/20 0.63
LMNA P02545 3/20 0.61
CYP1A2 P05177 2/20 0.61
NFKB1 P19838 2/20 0.61
ACHE P22303 2/20 0.61
PMP22 Q01453 2/20 0.61
ESR1 P03372 1/20 0.61
MAPT P10636 1/20 0.61
BLM P54132 1/20 0.61
SMN1; SMN2 Q16637 3/20 0.57
RXFP1 Q9HBX9 2/20 0.57
USP2 O75604 1/20 0.57
TNF P01375 1/20 0.57
TSHR P16473 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9682263 0.91 TRPA1 (0.68) TRPA1PDE4AADORA2BPDE4BPDE4C
SCHEMBL11611142 0.87 LMNA (0.58) TRPA1PDE4AADORA2BPDE4BPDE4C
SCHEMBL14985852 0.87 LMNA (0.58) TRPA1PDE4AADORA2BPDE4BPDE4C
SCHEMBL7989435 0.86 PDE4A (0.70) TRPA1PDE4AADORA2BPDE4BPDE4C
SCHEMBL5256903 0.86 PDE4A (0.70) TRPA1PDE4AADORA2BPDE4BPDE4C
SCHEMBL2924694 0.86 LMNA (0.60) TRPA1PDE4AADORA2BPDE4BPDE4C
SCHEMBL8697424 0.86 PDE4A (0.70) TRPA1PDE4AADORA2BPDE4BPDE4C
SCHEMBL11612265 0.86 PDE4A (0.64) TRPA1PDE4AADORA2BPDE4BPDE4C
SCHEMBL9297147 0.86 PDE4A (0.80) TRPA1PDE4AADORA2BPDE4BPDE4C
SCHEMBL10693536 0.86 PDE4A (0.71) TRPA1PDE4AADORA2BPDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5082845-A Gastrointestinal HOECHST JAPAN LIMITED (JP) 1992-01-21 US disclosed
EP-0330031-B1 THERAPEUTIC AGENTS FOR THE TREATMENT OF PEPTIC ULCER DISEASE HOECHST JAPAN LIMITED (JP) 1991-12-11 EP disclosed
EP-0330031-A1 Therapeutic agents for the treatment of peptic ulcer disease HOECHST JAPAN LIMITED (JP) 1989-08-30 EP disclosed