SCHEMBL10694210

SCHEMBL10694210

CC1(C)C(=O)N(Cc2ccccc2)c2cc3[nH]c(-c4ccncc4)nc3cc21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.51
PDE4B Q07343 1/20 0.51
PDE4C Q08493 1/20 0.51
PDE4D Q08499 1/20 0.51
PDE3B Q13370 1/20 0.51
PDE3A Q14432 1/20 0.51
AURKA O14965 1/20 0.46
AURKB Q96GD4 1/20 0.46
RHEB Q15382 1/20 0.44
ELANE P08246 1/20 0.42
ALDH1A1 P00352 5/20 0.41
HSD17B10 Q99714 3/20 0.41
KDM4E B2RXH2 3/20 0.41
HPGD P15428 3/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
PKN1 Q16512 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10696409 0.89 HPGD (0.50) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL10696080 0.87 TDP1 (0.50) AURKAAURKBALDH1A1HSD17B10KDM4E
SCHEMBL10696602 0.86 AURKA (0.60) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL10696040 0.85 AURKA (0.49) AURKAAURKBKDM4ENPC1MAPT
SCHEMBL10696033 0.85 PDE4A (0.54) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL10698598 0.84 PDE4A (0.53) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL10696394 0.83 PDE4A (0.52) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL10698025 0.82 PDE4A (0.51) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL10693690 0.82 PDE4A (0.51) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL10532292 0.82 PDE4A (0.48) PDE4APDE4BPDE4CPDE4DPDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0268178-A1 Pyrrolo-benzimidazoles, medicaments containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-05-25 EP disclosed