SCHEMBL10694966

SCHEMBL10694966

CC(=O)CCn1c(=O)[nH]c2ncn(CC(C)=O)c2c1=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 4/20 0.48
PDE4B Q07343 3/20 0.48
PDE4C Q08493 3/20 0.48
PDE4D Q08499 3/20 0.48
ADORA2B P29275 2/20 0.48
ADORA2A P29274 1/20 0.48
CNOT7 Q9UIV1 9/20 0.44
TRPA1 O75762 1/20 0.44
PARN O95453 1/20 0.43
LMNA P02545 2/20 0.40
MAPT P10636 2/20 0.40
BLM P54132 2/20 0.40
PMP22 Q01453 2/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP3A4 P08684 1/20 0.40
TSHR P16473 1/20 0.40
ESR1 P03372 1/20 0.40
CYP1A2 P05177 1/20 0.40
NFKB1 P19838 1/20 0.40
ACHE P22303 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21861608 0.91 TRPA1 (0.53) PDE4APDE4BPDE4CPDE4DADORA2B
SCHEMBL10696644 0.88 ADORA2B (0.65) PDE4APDE4BPDE4CPDE4DADORA2B
SCHEMBL10696193 0.86 PDE4A (0.46) PDE4APDE4BPDE4CPDE4DADORA2B
SCHEMBL11078954 0.82 ADORA2B (0.48) PDE4APDE4BPDE4CPDE4DADORA2B
SCHEMBL21861597 0.82 TRPA1 (0.59) PDE4APDE4BPDE4CPDE4DADORA2B
SCHEMBL9350776 0.81 PDE4A (0.43) PDE4APDE4BPDE4CPDE4DADORA2B
SCHEMBL9350658 0.80 CNOT7 (0.43) PDE4APDE4BPDE4CPDE4DCNOT7
SCHEMBL10696123 0.77 PDE4A (0.76) PDE4APDE4BPDE4CPDE4DADORA2B
SCHEMBL661486 0.76 CNOT7 (0.47) PDE4APDE4BPDE4CPDE4DADORA2B
SCHEMBL7318570 0.75 GDA (0.55) PDE4APDE4BPDE4CPDE4DADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0260127-A2 Xanthine derivatives, their preparation and pharmaceutical compositions containing them BEECHAM - WUELFING GmbH & Co. KG (DE) 1988-03-16 EP disclosed