SCHEMBL10695073

SCHEMBL10695073

CC(=O)Nc1ccc2c(c1)CC(=O)N2C

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.55
POLB P06746 2/20 0.55
MAOA P21397 3/20 0.52
TRIM24 O15164 1/20 0.50
PKM P14618 2/20 0.49
CYP1A2 P05177 1/20 0.49
ADRA2A P08913 1/20 0.49
SLC6A2 P23975 1/20 0.49
HTR2C P28335 1/20 0.49
SLC6A4 P31645 1/20 0.49
HTR2B P41595 1/20 0.49
HSP90AA1 P07900 1/20 0.48
TLR9 Q9NR96 1/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
MAPT P10636 2/20 0.48
MEN1 O00255 1/20 0.48
KDM4A O75164 1/20 0.48
THRB P10828 1/20 0.48
RECQL P46063 1/20 0.48
KMT2A Q03164 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24430173 0.82 NPC1 (0.53) ALDH1A1POLBTRIM24PKMSMN1; SMN2
SCHEMBL24430193 0.82 PKM (0.59) ALDH1A1POLBTRIM24PKMSLC6A2
SCHEMBL10508408 0.81 ALDH1A1 (0.47) ALDH1A1POLBMAOACYP1A2ADRA2A
SCHEMBL24430192 0.81 EPHX1 (0.56) ALDH1A1POLBPKMCYP1A2SLC6A2
SCHEMBL23055895 0.81 TRIM24 (0.54) ALDH1A1POLBTRIM24PKMMEN1
SCHEMBL19357202 0.80 MAPT (0.60) ALDH1A1TRIM24PKMMAPTMEN1
SCHEMBL24430169 0.77 MAPT (0.68) ALDH1A1SMN1; SMN2MAPTMEN1KMT2A
SCHEMBL19674328 0.77 TRIM24 (0.51) ALDH1A1POLBTRIM24PKMMEN1
SCHEMBL19669652 0.75 CYP1A2 (0.52) ALDH1A1POLBMAOACYP1A2SMN1; SMN2
SCHEMBL27940529 0.74 HDAC1 (0.50) ALDH1A1HSP90AA1TLR9MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103554008-A 1,3-substituted-5-acetaminoindolone compounds and application thereof to anti-tumor drugs UNIV TIANJIN SCIENCE & TECH 2014-02-05 CN disclosed
EP-0268178-A1 Pyrrolo-benzimidazoles, medicaments containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-05-25 EP disclosed