SCHEMBL19669652

SCHEMBL19669652

CC(=O)Nc1ccc2c(c1)OCC(=O)N2C

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.52
CYP2C19 P33261 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
POLB P06746 2/20 0.49
ALDH1A1 P00352 1/20 0.49
MAPT P10636 3/20 0.49
MAOA P21397 2/20 0.49
CYP11B1 P15538 1/20 0.47
CYP11B2 P19099 1/20 0.47
AAK1 Q2M2I8 1/20 0.46
IDH1 O75874 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.44
TP53 P04637 1/20 0.44
HSD17B10 Q99714 1/20 0.44
GABRG2 P18507 1/20 0.44
GABRB3 P28472 1/20 0.44
GABRA5 P31644 1/20 0.44
SYK P43405 1/20 0.43
TSHR P16473 1/20 0.43
CHRNB4 P30926 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19669631 0.83 RORC (0.57) CYP1A2CYP2C19NPSR1POLBALDH1A1
SCHEMBL21893436 0.82 CYP11B2 (0.51) CYP11B1CYP11B2IDH1GABRG2GABRB3
SCHEMBL8146771 0.81 CYP11B2 (0.50) MAPTCYP11B1CYP11B2GABRA5PDE3B
SCHEMBL19669650 0.80 NOS3 (0.51) CYP1A2CYP2C19NPSR1POLBALDH1A1
SCHEMBL19669654 0.80 TSHR (0.51) CYP1A2CYP2C19NPSR1POLBALDH1A1
SCHEMBL19669648 0.79 TSHR (0.45) CYP1A2CYP2C19NPSR1POLBALDH1A1
SCHEMBL19669633 0.79 CYP3A4 (0.52) CYP1A2CYP2C19NPSR1POLBMAPT
SCHEMBL19669647 0.78 ITGB3 (0.63)
SCHEMBL6532124 0.78 NPC1 (0.60) POLBALDH1A1MAPTMAOASMN1; SMN2
SCHEMBL17479101 0.76 RAB9A (0.48) NPSR1POLBALDH1A1MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9834520-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2017-12-05 US disclosed