SCHEMBL10695550

SCHEMBL10695550

CC1C(=O)N(C)c2cc3c(cc21)nc(-c1ccncc1)n3C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
ATM Q13315 1/20 0.39
PDE3B Q13370 3/20 0.37
PDE3A Q14432 3/20 0.37
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA9 Q16790 1/20 0.36
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
DHFR P00374 1/20 0.35
KDM4E B2RXH2 1/20 0.34
NPC1 O15118 1/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
TP53 P04637 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10696064 0.95 MEN1 (0.47) MEN1KMT2AATMPDE3BPDE3A
SCHEMBL10694972 0.87 MEN1 (0.40) MEN1KMT2ACA12CA1CA2
SCHEMBL10699478 0.84 MEN1 (0.41) MEN1KMT2AATMPDE3BPDE3A
SCHEMBL10699875 0.82 MEN1 (0.40) MEN1KMT2AATMPDE3BPDE3A
SCHEMBL10695521 0.81 CYP11B2 (0.53) ATMCYP11B1CYP11B2DHFRKIT
SCHEMBL10695097 0.80 PARP1 (0.40) MEN1KMT2ACA12CA1CA2
SCHEMBL10701679 0.80 MEN1 (0.41) MEN1KMT2AATMPDE3BPDE3A
SCHEMBL10699877 0.79 MEN1 (0.41) MEN1KMT2AATMPDE3BPDE3A
SCHEMBL10694340 0.75 CA12 (0.50) MEN1KMT2ACA12CA9DHFR
SCHEMBL10694143 0.75 ALDH1A1 (0.48) ATMPDE3BPDE3AKDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0268178-A1 Pyrrolo-benzimidazoles, medicaments containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-05-25 EP disclosed