SCHEMBL10695729

SCHEMBL10695729

COc1ccc(-c2nc3cc4c(cc3[nH]2)N(C)C(=O)C4C)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB11 O95342 1/20 0.48
MAOA P21397 1/20 0.48
ADORA2A P29274 1/20 0.48
PDE3B Q13370 1/20 0.48
PDE3A Q14432 1/20 0.48
SLC2A1 P11166 1/20 0.48
NPC1 O15118 5/20 0.47
SMN1; SMN2 Q16637 5/20 0.47
RAB9A P51151 4/20 0.47
MAPT P10636 3/20 0.47
MEN1 O00255 2/20 0.47
LMNA P02545 2/20 0.47
KMT2A Q03164 2/20 0.47
NFKB1 P19838 2/20 0.47
NFKB2 Q00653 2/20 0.47
RELA Q04206 2/20 0.47
GAA P10253 1/20 0.47
MAPK1 P28482 1/20 0.47
STAT1 P42224 1/20 0.47
HTT P42858 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10696182 0.86 SCD (0.46) ADORA2ASMN1; SMN2NPBWR1ALDH1A1HPGD
SCHEMBL10700351 0.86 SLC2A1 (0.46) ABCB11MAOAADORA2APDE3BPDE3A
SCHEMBL10699596 0.86 SLC2A1 (0.46) ABCB11MAOAADORA2APDE3BPDE3A
SCHEMBL10694143 0.85 ALDH1A1 (0.48) PDE3BPDE3ANPC1RAB9AMAPT
SCHEMBL2492174 0.83 SLC2A1 (0.46) ABCB11MAOAADORA2APDE3BPDE3A
SCHEMBL10530486 0.80 ABCB11 (0.46) ABCB11MAOAADORA2APDE3BPDE3A
SCHEMBL10695474 0.79 MAPT (0.54) NPC1SMN1; SMN2RAB9AMAPTKMT2A
SCHEMBL10699168 0.76 SLC2A1 (0.49) ABCB11MAOAADORA2APDE3BPDE3A
SCHEMBL10695270 0.76 NPC1 (0.50) ABCB11MAOAADORA2APDE3BPDE3A
SCHEMBL10696060 0.76 CBFB (0.54) NPC1SMN1; SMN2RAB9AMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0268178-A1 Pyrrolo-benzimidazoles, medicaments containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-05-25 EP disclosed