SCHEMBL10697748

SCHEMBL10697748

CC(C(=O)O)c1cc(Br)ccc1N

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.50
GLA P06280 1/20 0.50
MAPT P10636 3/20 0.45
POLB P06746 1/20 0.45
GAA P10253 1/20 0.45
PLAU P00749 1/20 0.40
HDAC1 Q13547 1/20 0.39
NPC1 O15118 1/20 0.38
MAPK1 P28482 1/20 0.38
HTT P42858 1/20 0.38
PTGS2 P35354 8/20 0.38
PTGS1 P23219 6/20 0.38
HPGD P15428 1/20 0.37
LMNA P02545 2/20 0.36
CYP2C9 P11712 2/20 0.36
AKR1C3 P42330 2/20 0.36
CXCR1 P25024 2/20 0.36
CXCR2 P25025 2/20 0.36
ALB P02768 1/20 0.36
ESR1 P03372 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27603483 0.87 KDM4E (0.47) KDM4EGLAMAPTPOLBGAA
SCHEMBL38661512 0.86 KDM4E (0.46) KDM4EGLAMAPTPOLBGAA
SCHEMBL3180180 0.80 TDP1 (0.40) POLBHTTPTGS2PTGS1HPGD
SCHEMBL8324702 0.80 PTGS1 (0.57) KDM4EMAPTPOLBGAAHTT
SCHEMBL3984863 0.77 KDM4E (0.42) KDM4EGLAMAPTPOLBGAA
SCHEMBL283021 0.77 GABRA1 (0.46) KDM4EGLAMAPTPOLBGAA
SCHEMBL8157598 0.76 GRM1 (0.41) HTTPTGS2PTGS1LMNAPPARA
SCHEMBL1678995 0.76 GRM1 (0.41) HTTPTGS2PTGS1LMNAPPARA
SCHEMBL16293581 0.76 PTGS1 (0.60) KDM4EMAPTPOLBPTGS2PTGS1
SCHEMBL16293535 0.76 PTGS1 (0.60) KDM4EMAPTPOLBPTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0255178-A2 Process for preparing hetero aryl and aryl alkanoic acids Nobel Chemicals AB (SE) 1988-02-03 EP disclosed