SCHEMBL8324702

SCHEMBL8324702

CC(C(=O)O)c1cc(Br)ccc1O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.57
PTGS2 P35354 1/20 0.57
HPGD P15428 4/20 0.50
ALOX15 P16050 2/20 0.46
CES2 O00748 1/20 0.46
GALR3 O60755 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2C9 P11712 1/20 0.46
CASP1 P29466 1/20 0.46
CYP2C19 P33261 1/20 0.46
NPSR1 Q6W5P4 3/20 0.45
LMNA P02545 2/20 0.45
MAPT P10636 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
KMT2A Q03164 4/20 0.43
MEN1 O00255 3/20 0.43
POLB P06746 2/20 0.43
L3MBTL1 Q9Y468 2/20 0.42
TP53 P04637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27506947 0.87 HPGD (0.48) PTGS1PTGS2HPGDALOX15CES2
SCHEMBL3180180 0.81 TDP1 (0.40) PTGS1PTGS2HPGDLMNATDP1
SCHEMBL490883 0.81 PTGS2 (0.60) PTGS1PTGS2ALOX15CES2CYP1A2
SCHEMBL9744811 0.81 HPGD (0.48) HPGDALOX15CES2GALR3CYP1A2
SCHEMBL8321938 0.81 HPGD (0.47) PTGS1PTGS2HPGDALOX15CES2
SCHEMBL10697748 0.80 KDM4E (0.50) PTGS1PTGS2HPGDCYP2C9LMNA
SCHEMBL31182212 0.78 GABRA1 (0.58) PTGS1HPGDALOX15CES2GALR3
SCHEMBL282835 0.78 GABRA1 (0.58) PTGS1HPGDALOX15CES2GALR3
SCHEMBL8157598 0.78 GRM1 (0.41) PTGS1PTGS2CYP1A2LMNATDP1
SCHEMBL6591473 0.78 PTGS2 (0.57) PTGS1PTGS2HPGDALOX15CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733033-B1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LTD (GB) 1999-12-22 EP disclosed
CN-1201454-A Meta-guanidino, ureido, thioureido or azacyclic aminobenzoic acid derivatives as integrin antagonists SEARLE & CO (US) 1998-12-09 CN disclosed
EP-0733033-A1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LIMITED (GB) 1996-09-25 EP disclosed
WO-1996011902-A1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LIMITED (GB) 1996-04-25 WO disclosed