SCHEMBL1069872

SCHEMBL1069872

FC(F)Oc1[c]cc(OC(F)(F)F)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR3 P46089 5/20 0.37
MAPT P10636 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.33
KIF11 P52732 1/20 0.33
KDM4E B2RXH2 1/20 0.33
EPHX2 P34913 1/20 0.33
ALDH1A1 P00352 1/20 0.32
PDE2A O00408 2/20 0.32
CES1 P23141 1/20 0.32
SCN5A Q14524 2/20 0.31
NPC1 O15118 2/20 0.31
LMNA P02545 2/20 0.31
RAB9A P51151 2/20 0.31
GMNN O75496 1/20 0.31
USP2 O75604 1/20 0.31
TP53 P04637 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
ADORA3 P0DMS8 1/20 0.31
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1064079 0.87 GPR3 (0.34) GPR3MAPTKIF11EPHX2ALDH1A1
SCHEMBL900696 0.85 DRD1 (0.38) MAPTKDM4EALDH1A1NPC1LMNA
SCHEMBL160011 0.78 GPR3 (0.35) GPR3MAPTL3MBTL1KIF11EPHX2
SCHEMBL1068998 0.75 GPR3 (0.37) GPR3KIF11PDE2ACES1SCN5A
SCHEMBL1067709 0.74 MEN1 (0.31) MAPTLMNASMN1; SMN2
SCHEMBL21268362 0.74 MAPT (0.34) GPR3MAPTL3MBTL1KDM4EEPHX2
SCHEMBL4915707 0.74 L3MBTL1 (0.44) GPR3L3MBTL1ALDH1A1PDE2ALMNA
SCHEMBL457425 0.73 GPR3 (0.37) GPR3MAPTL3MBTL1KIF11KDM4E
SCHEMBL28379631 0.73 EPHX2 (0.39) GPR3MAPTL3MBTL1KIF11KDM4E
SCHEMBL1069758 0.72 MAPT (0.37) MAPTKDM4EALDH1A1NPC1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436961-B1 SUBSTANCE P RECEPTOR ANTAGONIST; 2-PHENYL-3-BENZYLAMINOPIPERIDINES PFIZER INC 2002-08-20 US claimed
EP-2900645-B1 HERBICIDAL AND FUNGICIDAL 3-PHENYLISOXAZOLIN DERIVATIVES BAYER CROPSCIENCE AG (DE) 2019-08-21 EP disclosed
WO-2011006886-A2 AZOLE COMPOUNDS CARRYING A SULFUR SUBSTITUENT XIV BASF SE (DE) 2011-01-20 WO disclosed
WO-2010149758-A1 ANTIFUNGAL 1, 2, 4-TRIAZOLYL DERIVATIVES BASF SE (DE) 2010-12-29 WO disclosed
EP-1172106-A2 Use of fluoroalkoxybenzylamino derivatives of nitrogen containing heterocycles as substance P receptor antagonists Pfizer Products Inc. (US) 2002-01-16 EP disclosed