SCHEMBL10705671

SCHEMBL10705671

c1ccc(-c2ccc(CN3CC[N]CC3)cc2)cc1

nearest known ligand 0.64

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.59
TSHR P16473 1/20 0.59
CYP2D6 P10635 2/20 0.59
CYP2C19 P33261 1/20 0.59
CHKA P35790 1/20 0.57
SIGMAR1 Q99720 2/20 0.55
HRH3 Q9Y5N1 4/20 0.55
HRH4 Q9H3N8 1/20 0.55
KCNH2 Q12809 1/20 0.51
FAAH O00519 2/20 0.50
LMNA P02545 1/20 0.50
POLB P06746 1/20 0.50
MGLL Q99685 1/20 0.49
MAPK1 P28482 1/20 0.49
KMT2A Q03164 1/20 0.49
LSS P48449 1/20 0.49
HTR2B P41595 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL41501 0.88 SIGMAR1 (0.71) SIGMAR1LMNAPOLBKMT2A
SCHEMBL1111888 0.84 DRD4 (0.53) SIGMAR1HRH3FAAHMGLL
SCHEMBL16226080 0.84 SIGMAR1 (0.78) ALDH1A1TSHRCYP2D6CYP2C19CHKA
SCHEMBL1690956 0.82 CYP2D6 (0.85) ALDH1A1TSHRCYP2D6CYP2C19CHKA
SCHEMBL42218 0.81 SIGMAR1 (0.61) ALDH1A1CYP2D6CYP2C19SIGMAR1HRH3
SCHEMBL24023622 0.81 CYP2D6 (0.89) ALDH1A1CYP2D6CYP2C19CHKASIGMAR1
SCHEMBL1997330 0.81 CYP2D6 (0.89) ALDH1A1CYP2D6CYP2C19CHKASIGMAR1
SCHEMBL24023625 0.81 CYP2D6 (0.89) ALDH1A1CYP2D6CYP2C19CHKASIGMAR1
SCHEMBL1111800 0.80 HTR7 (0.60) HRH3FAAHMGLL
SCHEMBL27674930 0.79 CYP2D6 (0.61) ALDH1A1TSHRCYP2D6CYP2C19CHKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0284552-A1 4-Benzyl-piperazinyl-hydrazones CIBA-GEIGY AG (CH) 1988-09-28 EP claimed
EP-0284552-A1 4-Benzyl-piperazinyl-hydrazones CIBA-GEIGY AG (CH) 1988-09-28 EP disclosed