SCHEMBL10709133

SCHEMBL10709133

Nc1nc(N)c2ncn([C@]3(CC(c4ccccc4)c4ccc(Cl)cc4)O[C@H](CO)[C@@H](O)[C@H]3O)c2n1

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 9/20 0.42
ADORA2B P29275 8/20 0.42
ADORA1 P30542 5/20 0.42
ADORA3 P0DMS8 4/20 0.42
HINT1 P49773 1/20 0.40
CYP1A2 P05177 1/20 0.39
THPO P40225 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10707941 0.97 ADORA2A (0.42) ADORA2AADORA2BADORA1ADORA3HINT1
SCHEMBL10709115 0.95 ADORA2A (0.45) ADORA2AADORA2BADORA1ADORA3HINT1
SCHEMBL11015150 0.92 ADORA2A (0.41) ADORA2AADORA2BADORA1ADORA3HINT1
SCHEMBL10709057 0.90 ADORA2A (0.48) ADORA2AADORA2BADORA1ADORA3
SCHEMBL10711083 0.89 ADORA3 (0.45) ADORA2AADORA2BADORA1ADORA3
SCHEMBL10710910 0.87 ADORA2A (0.46) ADORA2AADORA2BADORA1ADORA3
SCHEMBL10707529 0.85 ADORA3 (0.47) ADORA2AADORA2BADORA1ADORA3
SCHEMBL3450684 0.83 ADORA3 (0.48) ADORA2AADORA2BADORA1ADORA3
SCHEMBL10709847 0.83 ADORA3 (0.43) ADORA2AADORA2BADORA1ADORA3
SCHEMBL10712341 0.81 ADORA3 (0.44) ADORA2AADORA2BADORA1ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0139358-B1 N6-SUBSTITUTED DIARYLALKYL ADENOSINES, PROCESSES FOR THEIR PRODUCTION AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME WARNER-LAMBERT COMPANY (US) 1988-11-09 EP disclosed
EP-0139358-A2 N6-substituted diarylalkyl adenosines, processes for their production and pharmaceutical compositions comprising the same WARNER-LAMBERT COMPANY (US) 1985-05-02 EP disclosed