SCHEMBL10731925

SCHEMBL10731925

CN1c2ccccc2C(c2ccco2)=NCC1CNC(=O)c1ccco1

nearest known ligand 0.57

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 7/20 0.54
OPRK1 P41145 7/20 0.52
OPRD1 P41143 5/20 0.52
OPRM1 P35372 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10737425 0.99 CCKBR (0.53) CCKBROPRK1OPRD1OPRM1
SCHEMBL11144787 0.90 OPRK1 (0.56) CCKBROPRK1OPRD1OPRM1
SCHEMBL11138033 0.89 CCKBR (0.69) CCKBROPRK1OPRD1OPRM1
SCHEMBL10732104 0.87 OPRK1 (0.54) CCKBROPRK1OPRD1OPRM1
Hydrochloric Acid SCHEMBL10730349 0.86 OPRK1 (0.53) CCKBROPRK1OPRD1OPRM1
SCHEMBL11137502 0.85 CCKBR (0.47) CCKBROPRK1OPRD1OPRM1
SCHEMBL11144159 0.80 OPRK1 (0.63) CCKBROPRK1OPRD1OPRM1
SCHEMBL10730756 0.80 CCKBR (0.41) CCKBROPRK1OPRD1OPRM1
Hydrochloric Acid SCHEMBL11145247 0.79 OPRK1 (0.62) CCKBROPRK1OPRD1OPRM1
SCHEMBL11139219 0.78 MTNR1A (0.46) CCKBROPRK1OPRD1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4649137-A ANALGESICS KALI-CHEMIE PHARMA GMBH (DE) 1987-03-10 US disclosed
EP-0068240-B1 2-ACYLAMINOMETHYL-1,4-BENZODIAZEPINE DERIVATIVES, THEIR PREPARATION AND INTERMEDIATES, AND PHARMACEUTICAL PREPARATIONS CONTAINING THEM Kali-Chemie Pharma GmbH (DE) 1985-09-25 EP disclosed
US-4497740-A ANALGESICS KALI-CHEMIE PHARMA GMBH (DE) 1985-02-05 US disclosed
EP-0068240-A1 2-Acylaminomethyl-1,4-benzodiazepine derivatives, their preparation and intermediates, and pharmaceutical preparations containing them Kali-Chemie Pharma GmbH (DE) 1983-01-05 EP disclosed