SCHEMBL107531

SCHEMBL107531

O=C(OCc1ccc(Cl)cc1)ON1CCN(CC[S+]([O-])c2ccc3[nH]c(=O)oc3c2)CC1

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 14/20 0.47
KCNH2 Q12809 2/20 0.47
ATXN2 Q99700 8/20 0.43
HTR1A P08908 1/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A3 Q01959 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL104877 0.93 ENPP2 (0.55) ENPP2KCNH2ATXN2
SCHEMBL104770 0.88 ENPP2 (0.61) ENPP2KCNH2ATXN2
SCHEMBL1671586 0.88 ENPP2 (0.48) ENPP2KCNH2ATXN2
SCHEMBL1670435 0.86 ENPP2 (0.43) ENPP2KCNH2ATXN2HTR1ASLC6A2
SCHEMBL1672873 0.84 ENPP2 (0.42) ENPP2KCNH2ATXN2
SCHEMBL104876 0.81 ENPP2 (0.70) ENPP2KCNH2ATXN2
SCHEMBL13137773 0.81 ENPP2 (0.70) ENPP2KCNH2ATXN2
SCHEMBL13137772 0.81 ENPP2 (0.70) ENPP2KCNH2ATXN2
SCHEMBL6162014 0.78 GRIN1 (0.54)
SCHEMBL103926 0.78 ENPP2 (0.48) ENPP2KCNH2ATXN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2426106-B1 Piperidine and Piperazine derivatives for the treatment of tumours MERCK PATENT GMBH (DE) 2013-07-31 EP disclosed
EP-2426106-A1 Piperidine and Piperazine derivatives for the treatment of tumours Merck Patent GmbH (DE) 2012-03-07 EP disclosed