SCHEMBL1672873

SCHEMBL1672873

O=C(OCc1cc(F)cc(C(F)(F)F)c1)ON1CCN(CC[S+]([O-])c2ccc3[nH]c(=O)oc3c2)CC1

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 14/20 0.42
ATXN2 Q99700 9/20 0.42
KCNH2 Q12809 2/20 0.42
GRIN2D O15399 2/20 0.36
GRIN3B O60391 2/20 0.36
GRIN1 Q05586 2/20 0.36
GRIN2A Q12879 2/20 0.36
GRIN2B Q13224 2/20 0.36
GRIN2C Q14957 2/20 0.36
GRIN3A Q8TCU5 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1671586 0.93 ENPP2 (0.48) ENPP2ATXN2KCNH2
SCHEMBL11898731 0.90 ENPP2 (0.53) ENPP2ATXN2KCNH2
SCHEMBL11898730 0.90 ENPP2 (0.53) ENPP2ATXN2KCNH2
SCHEMBL104877 0.86 ENPP2 (0.55) ENPP2ATXN2KCNH2
SCHEMBL107531 0.84 ENPP2 (0.47) ENPP2ATXN2KCNH2
SCHEMBL1670435 0.84 ENPP2 (0.43) ENPP2ATXN2KCNH2GRIN2DGRIN3B
SCHEMBL11899032 0.82 ENPP2 (0.60) ENPP2ATXN2KCNH2
SCHEMBL11899033 0.82 ENPP2 (0.60) ENPP2ATXN2KCNH2
SCHEMBL15304438 0.80 ENPP2 (0.55) ENPP2ATXN2KCNH2
SCHEMBL1671516 0.77 ENPP2 (0.35) ENPP2ATXN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2488504-B1 SULFOXIDE DERIVATIVES FOR TREATING TUMORS MERCK PATENT GMBH (DE) 2016-07-06 EP disclosed
EP-2488504-A1 SULFOXIDE DERIVATIVES FOR TREATING TUMORS Merck Patent GmbH (DE) 2012-08-22 EP disclosed
WO-2011044978-A1 SULFOXIDE DERIVATIVES FOR TREATING TUMORS MERCK PATENT GMBH (DE) 2011-04-21 WO disclosed