SCHEMBL1075769

SCHEMBL1075769

CC(C)Cc1nc(Br)c(Br)[nH]1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.41
KDM4E B2RXH2 1/20 0.38
MAPT P10636 1/20 0.38
GSK3B P49841 1/20 0.36
ADORA3 P0DMS8 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA2B P29275 1/20 0.34
ADORA1 P30542 1/20 0.34
CCNE2 O96020 1/20 0.31
CCNE1 P24864 1/20 0.31
CDK2 P24941 1/20 0.31
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19402606 0.76 TSHR (0.36) TSHRKDM4EMAPTGSK3BADORA3
SCHEMBL19402609 0.76 TSHR (0.36) TSHRKDM4EMAPTGSK3BADORA3
SCHEMBL8807973 0.69 KDM4E (0.48) TSHRKDM4EMAPTGSK3BADORA3
SCHEMBL31546962 0.68 TSHR (0.43) TSHRKDM4EMAPTGSK3B
SCHEMBL12461900 0.67 TAAR1 (0.35)
SCHEMBL19402604 0.65 TSHR (0.41) TSHRKDM4EMAPTGSK3BADORA3
SCHEMBL13833511 0.64 TSHR (0.59) TSHRKDM4EMAPTGSK3BADORA3
SCHEMBL4105591 0.61 MGAM (0.46) KDM4EMAPT
SCHEMBL6756153 0.61 KDM4E (0.44) TSHRKDM4EMAPTGSK3BADORA3
SCHEMBL4053441 0.60 ADORA3 (0.40) TSHRKDM4EMAPTGSK3BADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2274300-A2 NOVEL HETEROCYCLIC COMPOUNDS AND USES THEROF Novartis AG (CH) 2011-01-19 EP disclosed
WO-2009115572-A2 NOVEL HETEROCYCLIC COMPOUNDS AND USES THEROF NOVARTIS AG (CH) 2009-09-24 WO disclosed