SCHEMBL10758604

SCHEMBL10758604

CO[C@@H]1C[C@H](OCc2ccccc2)[C@H](O)[C@@H](COC(c2ccccc2)(c2ccccc2)c2ccccc2)O1

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 1/20 0.38
TYMP P19971 14/20 0.38
PSEN1 P49768 1/20 0.35
PSEN2 P49810 1/20 0.35
APH1B Q8WW43 1/20 0.35
NCSTN Q92542 1/20 0.35
APH1A Q96BI3 1/20 0.35
PSENEN Q9NZ42 1/20 0.35
SLC6A2 P23975 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10758609 1.00 PDE4D (0.38) PDE4DTYMPPSEN1PSEN2APH1B
SCHEMBL10423649 0.91 PDE4D (0.38) PDE4DTYMPPSEN1PSEN2APH1B
SCHEMBL10423648 0.91 PDE4D (0.38) PDE4DTYMPPSEN1PSEN2APH1B
SCHEMBL19891704 0.85 PDE4D (0.49) PDE4DPSEN1PSEN2APH1BNCSTN
SCHEMBL10423644 0.85 TYMP (0.38) PDE4DTYMPPSEN1PSEN2APH1B
SCHEMBL10423643 0.85 TYMP (0.38) PDE4DTYMPPSEN1PSEN2APH1B
SCHEMBL9307935 0.83 TYMP (0.41) TYMP
SCHEMBL1776371 0.83 PDE4D (0.51) PDE4DPSEN1PSEN2APH1BNCSTN
SCHEMBL10755806 0.83 PDE4D (0.51) PDE4DPSEN1PSEN2APH1BNCSTN
SCHEMBL9307929 0.83 TYMP (0.41) TYMP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4683314-A ANTICHOLESTEROL MERCK & CO., INC. (US) 1987-07-28 US disclosed
US-4540796-A PREPARATION OF 4-HYDROXY-3,4,5,6-TETRAHYDRO-2H-PYRAN-2-ONE DERIVATIVE MERCK & CO., INC. (US) 1985-09-10 US disclosed
US-4440927-A Process for preparing inhibitors of 3-hydroxy-3-methylglutaryl coenzyme A reductase via a chiral synthon MERCK & CO., INC. (US) 1984-04-03 US disclosed