SCHEMBL1076367

SCHEMBL1076367

COc1c(NC2=NC(CC3CCOCC3)N=C2C)cccc1-c1ccccc1

nearest known ligand 0.33

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.33
KDM4E B2RXH2 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
CHRM3 P20309 6/20 0.33
JAK2 O60674 2/20 0.33
TTK P33981 1/20 0.33
JAK1 P23458 1/20 0.33
TYK2 P29597 1/20 0.33
PDCD1 Q15116 2/20 0.32
CD274 Q9NZQ7 2/20 0.32
MAPT P10636 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
PDE9A O76083 2/20 0.31
ITGB1 P05556 1/20 0.31
ITGA4 P13612 1/20 0.31
KCNH3 Q9ULD8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1075785 0.82 TTK (0.34) ALDH1A1KDM4EL3MBTL1CHRM3JAK2
SCHEMBL946112 0.76 ALDH1A1 (0.38) ALDH1A1KDM4EL3MBTL1JAK2JAK1
SCHEMBL946600 0.72 TTK (0.33) ALDH1A1KDM4EL3MBTL1JAK2TTK
SCHEMBL1076368 0.66 BACE1 (0.43)
SCHEMBL1075786 0.61 BACE1 (0.58)
Hydrochloric Acid SCHEMBL28181585 0.60 ALDH1A1 (0.43) ALDH1A1KDM4EL3MBTL1JAK2JAK1
SCHEMBL13385087 0.60 PDE4B (0.48) ALDH1A1KDM4EL3MBTL1PDCD1CD274
SCHEMBL3296653 0.59 ALDH1A1 (0.48) ALDH1A1KDM4EL3MBTL1PDCD1CD274
SCHEMBL5609138 0.58 PDE4B (0.36) KDM4EJAK2JAK1TYK2
SCHEMBL14176639 0.58 SCN8A (0.45) ALDH1A1KDM4EPDCD1CD274MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002408-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed