SCHEMBL10769486

SCHEMBL10769486

Cc1cc(C)c2nc([S+]([O-])Cc3cn4ccccc4n3)[nH]c2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.42
NPC1 O15118 5/20 0.42
RAB9A P51151 5/20 0.42
KDM4E B2RXH2 5/20 0.41
PKM P14618 3/20 0.41
TSHR P16473 2/20 0.38
SMN1; SMN2 Q16637 5/20 0.37
PDE10A Q9Y233 2/20 0.37
HTT P42858 1/20 0.37
MAPT P10636 4/20 0.37
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
DAPK3 O43293 1/20 0.36
ROCK2 O75116 1/20 0.36
PIM1 P11309 1/20 0.36
RPS6KB1 P23443 1/20 0.36
RPS6KA3 P51812 1/20 0.36
CSNK2A1 P68400 1/20 0.36
DYRK1A Q13627 1/20 0.36
PIM3 Q86V86 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10666860 0.80 NPC1 (0.57) KMT2ANPC1RAB9AKDM4EPKM
SCHEMBL6442937 0.78 CYP3A4 (0.40) NPC1RAB9AKDM4EPKMSMN1; SMN2
SCHEMBL6483036 0.77 NPC1 (0.64) KMT2ANPC1RAB9AKDM4EPKM
SCHEMBL6475549 0.74 NOS2 (0.38) RPS6KA3ESR1
SCHEMBL10617498 0.69 ESR1 (0.34) ESR1
SCHEMBL10617565 0.67 ADORA3 (0.44) KMT2ANPC1RAB9AKDM4EPDE10A
SCHEMBL6880563 0.63 CBFB (0.51) ALDH1A1ESR1MAPK10
SCHEMBL423547 0.63 NPC1 (0.58) KMT2ANPC1RAB9AKDM4ETSHR
SCHEMBL22499408 0.62 NPC1 (0.51) KMT2ANPC1RAB9AKDM4ETSHR
SCHEMBL6475793 0.61 ATP4A (0.57) KMT2ANPC1RAB9AKDM4EPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0242341-A1 Benzimidazoles, process for their preparation and preparations containing same Aktiebolaget Hässle (SE) 1987-10-21 EP disclosed
WO-1987005021-A1 BENZIMIDAZOLES AND THEIR PHARMACEUTICAL USE Aktiebolaget Hässle (SE) 1987-08-27 WO disclosed