SCHEMBL10769887

SCHEMBL10769887

C[C@@H](N)C(=O)NCC#Cc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.54
LMNA P02545 1/20 0.49
SIGMAR1 Q99720 1/20 0.49
GRIK1 P39086 1/20 0.48
GRIK2 Q13002 1/20 0.48
KMT2A Q03164 1/20 0.45
TAAR1 Q96RJ0 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC2 Q92769 1/20 0.45
HDAC8 Q9BY41 1/20 0.45
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
THPO P40225 1/20 0.44
FFAR1 O14842 1/20 0.44
LTA4H P09960 1/20 0.43
CTRB1 P17538 2/20 0.43
BLM P54132 1/20 0.43
PMP22 Q01453 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10421314 1.00 HTR2A (0.54) HTR2ALMNASIGMAR1GRIK1GRIK2
SCHEMBL3524487 0.86 SIGMAR1 (0.51) HTR2ALMNASIGMAR1GRIK1GRIK2
SCHEMBL10769885 0.77 SIGMAR1 (0.53) HTR2ALMNASIGMAR1GRIK1GRIK2
SCHEMBL10421315 0.77 CYP1A2 (0.48) HTR2ALMNASIGMAR1GRIK1GRIK2
SCHEMBL402415 0.75 TAAR1 (0.69) LMNAKMT2ATAAR1CYP2C19FFAR1
SCHEMBL10421320 0.75 LMNA (0.42) HTR2ALMNASIGMAR1KMT2AFFAR1
SCHEMBL24814159 0.74 GRIK1 (0.56) HTR2ALMNAGRIK1GRIK2KMT2A
SCHEMBL29178391 0.74 GRIK1 (0.56) HTR2ALMNAGRIK1GRIK2KMT2A
SCHEMBL1790978 0.74 KMT2A (0.63) KMT2AHDAC1HDAC2HDAC8CYP3A4
SCHEMBL2236118 0.74 KMT2A (0.63) KMT2AHDAC1HDAC2HDAC8CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0215297-A2 Substituted dipeptide amides G.D. Searle & Co. (US) 1987-03-25 EP disclosed