SCHEMBL10774385

SCHEMBL10774385

CC(C)C1(c2ccccc2OCCCCN2CCC(C(=O)c3ccc(F)cc3)CC2)Sc2ccccc2N(C)C1=O

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.51
CYP2D6 P10635 2/20 0.51
CYP2C9 P11712 1/20 0.51
NFKB1 P19838 1/20 0.51
THPO P40225 1/20 0.51
HIF1A Q16665 1/20 0.51
MEN1 O00255 1/20 0.51
GMNN O75496 1/20 0.51
LMNA P02545 1/20 0.51
MAPK1 P28482 1/20 0.51
BLM P54132 1/20 0.51
PMP22 Q01453 1/20 0.51
KMT2A Q03164 1/20 0.51
KDM4E B2RXH2 1/20 0.47
CYP1A2 P05177 1/20 0.47
HTR2A P28223 1/20 0.47
DRD2 P14416 1/20 0.44
HTR1A P08908 1/20 0.41
HTR7 P34969 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10770978 0.82 DRD2 (0.40) MEN1MAPK1KMT2AKDM4EHTR2A
Hydrochloric Acid SCHEMBL10570034 0.77 MEN1 (0.38) CYP3A4CYP2D6CYP2C9NFKB1THPO
SCHEMBL10771892 0.77 LMNA (0.53) LMNAKDM4E
Hydrochloric Acid SCHEMBL10772441 0.77 LMNA (0.44) CYP3A4CYP2D6CYP2C9NFKB1MEN1
SCHEMBL10710825 0.76 KDM4E (0.40) MEN1KMT2AKDM4EDRD2
Hydrochloric Acid SCHEMBL9829515 0.76 KMT2A (0.40) CYP3A4CYP2D6CYP2C9NFKB1THPO
Hydrochloric Acid SCHEMBL10770827 0.75 MEN1 (0.35) CYP3A4CYP2D6CYP2C9NFKB1THPO
Iprotiazem SCHEMBL10855448 0.75 HTR1A (0.40) MEN1KMT2AKDM4EDRD2HTR1A
Iprotiazem SCHEMBL2110235 0.75 HTR1A (0.40) MEN1KMT2AKDM4EDRD2HTR1A
Hydrochloric Acid SCHEMBL10573477 0.74 ABCB1 (0.39) CYP3A4CYP2D6CYP2C9MEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0244723-A2 Benzothiazinone derivatives, process for their preparation, medicaments containing them and their use HOECHST AKTIENGESELLSCHAFT (DE) 1987-11-11 EP disclosed