SCHEMBL1077648

SCHEMBL1077648

Cn1cc(OC(=O)Nc2ccc(F)cc2-c2ccc(Cl)c(F)c2)c(C(F)(F)F)n1

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 18/20 0.50
LMNA P02545 1/20 0.42
CHRM2 P08172 6/20 0.42
CHRM1 P11229 6/20 0.42
MAPT P10636 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1039642 0.94 CHRM3 (0.51) CHRM3LMNACHRM2CHRM1
SCHEMBL1039851 0.91 CHRM3 (0.43) CHRM3LMNAMAPTNPSR1
SCHEMBL3036773 0.86 CHRM3 (0.43) CHRM3LMNACHRM2CHRM1MAPT
SCHEMBL1078423 0.85 CHRM3 (0.50) CHRM3CHRM2CHRM1
SCHEMBL4835285 0.85 LMNA (0.39) CHRM3LMNACHRM2CHRM1NPSR1
SCHEMBL29505154 0.84 LMNA (0.53) CHRM3LMNAMAPTNPSR1
SCHEMBL302660 0.84 LMNA (0.53) CHRM3LMNAMAPTNPSR1
SCHEMBL5624615 0.83 CHRM3 (0.41) CHRM3LMNAMAPTNPSR1
SCHEMBL4848046 0.83 CHRM3 (0.48) CHRM3LMNACHRM2CHRM1MAPT
SCHEMBL3150885 0.82 CHRM3 (0.48) CHRM3LMNAMAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 46 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009071419-A1 FUNGICIDAL MIXTURES BASF SE (DE) 2009-06-11 WO claimed
WO-2009071389-A1 FUNGICIDE MIXTURES BASF SE (DE) 2009-06-11 WO claimed
WO-2009071450-A1 FUNGICIDAL MIXTURE BASF SE (DE) 2009-06-11 WO claimed
EP-2094080-B1 UTILISATION OF BLOCK COPOLYMERS BASED ON VINYL LACTAMES AND VINYL ACETATE AS SOLUBILISERS BASF SE (DE) 2017-06-07 EP disclosed
EP-2381770-B1 GEL FORMULA WHICH CAN BE STORED SAFELY FOR A LONG PERIOD WITH AT LEAST TWO ESSENTIALLY UNMIXED HYDROGELS BASF SE (DE) 2016-03-30 EP disclosed
EP-2271697-B1 ALCOHOL ALKOXYLATES, MEDIA CONTAINING THESE AND UTILISATION OF ALCOHOL ALKOXYLATES AS ADJUVANTS FOR THE AGROCHEMICAL SECTOR BASF SE (DE) 2014-07-09 EP disclosed
EP-2381770-A2 GEL FORMULATIONS THAT ARE STABLE FOR STORAGE, COMPRISING AT LEAST TWO SUBSTANTIALLY UN-MIXED HYDROGELS BASF SE (DE) 2011-11-02 EP disclosed
EP-2046784-B1 AZOLYLMETHYLOXIRANES, USE THEREOF FOR CONTROLLING PLANT PATHOGENIC FUNGI, AND AGENTS CONTAINING THE SAME BASF SE (DE) 2011-09-14 EP disclosed
EP-2069413-B1 ACTIVE INGREDIENT FORMULATIONS CONTAINING COMB POLYMERS BASF SE (DE) 2011-08-03 EP disclosed
EP-2278877-A2 CYCLODEXTRIN-CONTAINING SUSPENSION CONCENTRATES, METHOD FOR PRODUCING THE SAME AND THEIR USE BASF SE (DE) 2011-02-02 EP disclosed
EP-2041125-B1 AZOLYLMETHYLOXIRANES, THEIR USE FOR CONTROLLING PHYTOPATHOGENIC FUNGI AND AGENTS CONTAINING SAID COMPOUNDS BASF SE (DE) 2011-01-26 EP disclosed
WO-2008040786-A1 COMB POLYMERS AND USE THEREOF FOR THE PRODUCTION OF ACTIVE OR EFFECTIVE INGREDIENT FORMULATIONS BASF SE (DE) 2008-04-10 WO disclosed
WO-2008037607-A1 HETEROCYCLIC COMPOUNDS CONTAINING CARBONYL GROUPS, AND THE USE THEREOF FOR CONTROLLING PHYTOPATHOGENIC FUNGI BASF SE (DE) 2008-04-03 WO disclosed
WO-2008012246-A1 AZOLYLMETHYLOXIRANES, USE THEREOF FOR CONTROLLING PLANT PATHOGENIC FUNGI, AND AGENTS CONTAINING THE SAME BASF SE (DE) 2008-01-31 WO disclosed
WO-2008012234-A2 AZOLYLMETHYLOXIRANES, USE THEREOF FOR CONTROLLING PLANT PATHOGENIC FUNGI, AND AGENTS CONTAINING THE SAME BASF SE (DE) 2008-01-31 WO disclosed
WO-2008003607-A1 AZOLYLMETHYLOXIRANES, THEIR USE FOR CONTROLLING PHYTOPATHOGENIC FUNGI AND AGENTS CONTAINING SAID COMPOUNDS BASF SE (DE) 2008-01-10 WO disclosed
WO-2008003622-A1 AZOLYLMETHYLOXIRANES, THEIR USE FOR CONTROLLING PHYTOPATHOGENIC FUNGI AND AGENTS CONTAINING SAID COMPOUNDS BASF SE (DE) 2008-01-10 WO disclosed
WO-2007113136-A1 USE OF SUBSTITUTED TRIAZOLOPYRIMIDINES FOR CONTROLLING PHYTOPATHOGENIC HARMFUL FUNGI BASF AKTIENGESELLSCHAFT (DE) 2007-10-11 WO disclosed
WO-2007101810-A1 SUBSTITUTED TRIAZOLOPYRIMIDINES, METHODS FOR THE PRODUCTION THEREOF AND USE THEREOF FOR CONTROLLING PARASITIC FUNGI AND AGENTS CONTAINING THE SAME BASF SE (DE) 2007-09-13 WO disclosed
WO-2007101804-A1 SUBSTITUTED PYRAZOLOPYRIMIDINES, METHODS FOR THE PRODUCTION THEREOF AND USE THEREOF FOR CONTROLLING PARASITIC FUNGI AND AGENTS COMPRISING THE SAME BASF SE (DE) 2007-09-13 WO disclosed