SCHEMBL10778477

SCHEMBL10778477

O=C(O)c1cnc(-c2ccccc2)c2cc(F)ccc12

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 10/20 0.50
TDP1 Q9NUW8 2/20 0.48
CTDSP1 Q9GZU7 1/20 0.48
MAP2K4 P45985 1/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
MAP4K4 O95819 1/20 0.44
TAAR1 Q96RJ0 2/20 0.43
LDHA P00338 1/20 0.43
LMNA P02545 1/20 0.43
CYP1A2 P05177 1/20 0.43
MAPT P10636 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10782995 0.82 LDHA (0.47) DHODHMEN1KMT2ALDHALMNA
SCHEMBL10778479 0.79 TDP1 (0.45) DHODHTDP1CTDSP1MAP2K4TAAR1
SCHEMBL10783965 0.79 SMN1; SMN2 (0.53) DHODHTDP1MEN1KMT2ALDHA
SCHEMBL10781383 0.79 LDHA (0.56) DHODHMEN1KMT2ALDHALMNA
SCHEMBL9907710 0.73 HTR5A (0.52) MAP2K4LDHA
SCHEMBL11552012 0.72 DHODH (0.49) DHODHMEN1KMT2AMAP4K4LDHA
SCHEMBL15161302 0.72 MAP4K4 (0.81) DHODHMAP4K4
SCHEMBL5024503 0.71 LTB4R2 (0.51) DHODHMEN1KMT2ALMNAMAPT
SCHEMBL18573216 0.70 CNR1 (0.42) DHODHMEN1KMT2ALDHALMNA
SCHEMBL9907712 0.70 CSNK2A2 (0.52) MAP2K4MAP4K4LDHA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0105210-B1 ISOQUINOLINE DERIVATIVES, PROCESS FOR THEIR PREPARATION, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USE HOECHST AKTIENGESELLSCHAFT (DE) 1987-03-04 EP disclosed