SCHEMBL10779486

SCHEMBL10779486

CCC(C)(C(=O)O)c1ccc([N+](=O)[O-])c(F)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
ALDH1A1 P00352 4/20 0.40
HTT P42858 2/20 0.40
GAA P10253 1/20 0.40
THRB P10828 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
TTR P02766 1/20 0.39
APP P05067 1/20 0.38
NPC1 O15118 1/20 0.38
GLA P06280 1/20 0.38
MAPK1 P28482 1/20 0.38
CASP3 P42574 1/20 0.38
RAB9A P51151 1/20 0.38
SENP8 Q96LD8 1/20 0.38
SENP7 Q9BQF6 1/20 0.38
SENP6 Q9GZR1 1/20 0.38
TSHR P16473 1/20 0.37
HPD P32754 1/20 0.37
CASP6 P55212 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10779478 1.00 ATM (0.45) ATMTDP1ALDH1A1HTTGAA
SCHEMBL2527070 0.86 TSHR (0.53) ATMTDP1ALDH1A1HTTGAA
SCHEMBL112748 0.84 THRB (0.45) ATMTDP1ALDH1A1HTTGAA
SCHEMBL2531381 0.83 ALDH1A1 (0.40) TDP1ALDH1A1HTTGAANPC1
SCHEMBL1343471 0.83 TDP1 (0.45) ATMTDP1ALDH1A1HTTGAA
SCHEMBL5150306 0.83 TDP1 (0.45) ATMTDP1ALDH1A1HTTGAA
SCHEMBL3714548 0.82 ATM (0.50) ATMTDP1ALDH1A1HTTTTR
SCHEMBL3714543 0.82 ATM (0.50) ATMTDP1ALDH1A1HTTTTR
SCHEMBL28015054 0.82 ATM (0.39) ATMTDP1ALDH1A1HTTGAA
SCHEMBL11683508 0.82 MAPK1 (0.45) ALDH1A1HTTL3MBTL1NPC1GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0032620-B2 Process for preparing therapeutic 2-arylpropionic acids and esters, and novel arylmethylmalonate esters THE UPJOHN COMPANY (US) 1987-02-04 EP disclosed
EP-0032620-B1 Process for preparing therapeutic 2-arylpropionic acids and esters, and novel arylmethylmalonate esters THE UPJOHN COMPANY (US) 1984-05-30 EP disclosed
US-4398035-A INTERMEDIATE FOR FLURBIPROFEN THE UPJOHN COMPANY (US) 1983-08-09 US disclosed
US-4324904-A COMPOUND USEFUL IN MAKING FLURBIPROFEN THE UPJOHN COMPANY (US) 1982-04-13 US disclosed
EP-0032620-A1 Process for preparing therapeutic 2-arylpropionic acids and esters, and novel arylmethylmalonate esters THE UPJOHN COMPANY (US) 1981-07-29 EP disclosed