SCHEMBL10784304

SCHEMBL10784304

NC(=O)c1ccc(Cn2ccc(N)n2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
PARP10 Q53GL7 3/20 0.44
KMT2A Q03164 3/20 0.43
MEN1 O00255 2/20 0.43
KDM4E B2RXH2 2/20 0.43
PLA2G10 O15496 1/20 0.42
PLA2G2A P14555 1/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
LMNA P02545 2/20 0.42
CYP17A1 P05093 1/20 0.41
NNMT P40261 1/20 0.40
TSHR P16473 1/20 0.39
HTT P42858 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL184601 0.82 GAA (0.52) ALDH1A1TDP1KMT2AMEN1SMN1; SMN2
SCHEMBL12436753 0.80 LMNA (0.53) ALDH1A1TDP1KMT2AMEN1SMN1; SMN2
SCHEMBL10783151 0.78 LMNA (0.53) ALDH1A1KMT2AMEN1LMNATSHR
SCHEMBL1569200 0.78 ALDH1A1 (0.54) ALDH1A1L3MBTL1TDP1KMT2AMEN1
SCHEMBL1860285 0.76 ALDH1A1 (0.66) ALDH1A1L3MBTL1TDP1KMT2AMEN1
SCHEMBL17316533 0.76 ALDH1A1 (0.53) ALDH1A1L3MBTL1TDP1KMT2AMEN1
SCHEMBL17316607 0.76 ALDH1A1 (0.57) ALDH1A1L3MBTL1TDP1KMT2AMEN1
SCHEMBL2271144 0.76 L3MBTL1 (0.66) ALDH1A1L3MBTL1TDP1KMT2AMEN1
SCHEMBL3551388 0.76 HDAC1 (0.60) HDAC1
SCHEMBL634581 0.75 ALDH1A1 (0.65) ALDH1A1L3MBTL1TDP1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4665073-A HISTAMINE H2-ANTAGONISTS ICI AMERICAS INC. (GB) 1987-05-12 US disclosed
EP-0060094-B1 GUANIDINE DERIVATIVES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1986-01-22 EP disclosed
US-4447441-A ANTIHISTAMINE, ANTIULCER AND ANTISECRETORY AGENT IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1984-05-08 US disclosed
EP-0060094-A2 Guanidine derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1982-09-15 EP disclosed