Fenipentol

Fenipentol

SCHEMBL10795261

CC(=O)O.CCCCC(O)c1ccccc1

nearest known ligand 0.55

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADRA2AADRA2BADRA2CADRB2AGTR1AVPR1AAVPR1BAVPR2BDKRB2CALCRCHRNA3CHRNB4ESR1ESR2GHSRGNRHRGSC1HSPA8MALT1MC1RMC4RNOS1NOS2NOS3OPRK1OXTRRAMP1RAMP2RAMP3SCN5ASSTR1SSTR2SSTR3SSTR4SSTR5dacAdacBdacCfolPftsImrcAmrcBmrdArplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Fenipentol. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.55
KDM4E B2RXH2 1/20 0.55
LMNA P02545 2/20 0.55
ASAH1 Q13510 2/20 0.54
POLB P06746 1/20 0.53
RIPK1 Q13546 1/20 0.52
NPC1 O15118 2/20 0.51
RAB9A P51151 2/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
NAAA Q02083 2/20 0.49
CERT1 Q9Y5P4 3/20 0.48
CNR2 P34972 1/20 0.46
PPARG P37231 1/20 0.46
PPARA Q07869 1/20 0.46
ACER2 Q5QJU3 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fenipentol SCHEMBL11351770 0.92 LMNA (0.64) ALDH1A1KDM4ELMNAASAH1POLB
Fenipentol SCHEMBL21837 0.92 LMNA (0.64) ALDH1A1KDM4ELMNAASAH1POLB
Fenipentol SCHEMBL11573151 0.92 LMNA (0.64) ALDH1A1KDM4ELMNAASAH1POLB
Acetic Acid SCHEMBL29265549 0.90 LMNA (0.57) ALDH1A1KDM4ELMNAASAH1RIPK1
Acetic Acid SCHEMBL29265550 0.90 LMNA (0.57) ALDH1A1KDM4ELMNAASAH1RIPK1
Fenipentol SCHEMBL29913852 0.90 LMNA (0.61) ALDH1A1KDM4ELMNAASAH1POLB
Fenipentol SCHEMBL6535112 0.90 ALDH1A1 (0.50) ALDH1A1KDM4ELMNAASAH1POLB
Fenipentol SCHEMBL27583052 0.87 KDM4E (0.58) ALDH1A1KDM4ELMNAASAH1POLB
Fenipentol SCHEMBL27504649 0.86 LMNA (0.57) ALDH1A1KDM4ELMNAASAH1POLB
SCHEMBL28218362 0.86 LMNA (0.61) ALDH1A1KDM4ELMNAASAH1RIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4650898-A PERFUMES, FOODS, CHEWING GUMS INTERNATIONAL FLAVORS & FRAGRANCES INC. (US) 1987-03-17 US disclosed
US-4632831-A GRAFEFRUIT-LIKE INTERNATIONAL FLAVORS & FRAGRANCES INC. (US) 1986-12-30 US disclosed
US-4610812-A Uses of methyl phenyl pentanol derivatives in augmenting or enhancing the aroma or taste of consumable materials INTERNATIONAL FLAVORS & FRAGRANCES INC. (US) 1986-09-09 US disclosed