SCHEMBL10798232

SCHEMBL10798232

CCC(C(=O)c1c(F)cccc1F)n1cncn1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.45
PDE4D Q08499 1/20 0.41
CES2 O00748 2/20 0.39
CES1 P23141 2/20 0.39
KMT2A Q03164 2/20 0.37
HSP90AA1 P07900 1/20 0.37
CYP19A1 P11511 5/20 0.37
PDE4B Q07343 1/20 0.36
DPP8 Q6V1X1 2/20 0.35
DPP9 Q86TI2 2/20 0.35
DPP7 Q9UHL4 2/20 0.35
MEN1 O00255 1/20 0.34
PPARG P37231 1/20 0.34
PLAU P00749 1/20 0.33
ELANE P08246 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10799731 0.74 CYP19A1 (0.48) MAPTPDE4DKMT2AHSP90AA1CYP19A1
SCHEMBL5440264 0.73 MAPT (0.49) MAPTPDE4DKMT2AHSP90AA1CYP19A1
SCHEMBL10900677 0.71 MAPT (0.44) MAPTPDE4DKMT2AHSP90AA1CYP19A1
SCHEMBL2754295 0.71 MAPT (0.44) MAPTPDE4DKMT2AHSP90AA1CYP19A1
SCHEMBL21681423 0.70 KMT2A (0.34) MAPTPDE4DKMT2AHSP90AA1CYP19A1
SCHEMBL21681482 0.70 MAPT (0.38) MAPTPDE4DKMT2AHSP90AA1CYP19A1
SCHEMBL9748570 0.69 MAPT (0.63) MAPTPDE4DKMT2AHSP90AA1CYP19A1
SCHEMBL6319766 0.69 MAPT (0.44) MAPTKMT2AHSP90AA1CYP19A1
SCHEMBL22372311 0.68 CES2 (0.52) MAPTCES2CES1KMT2ADPP8
SCHEMBL11131956 0.68 JAK2 (0.39) MAPTKMT2AHSP90AA1CYP19A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0122693-B1 ANTIFUNGAL DI(AZOLYL)PROPANOL DERIVATIVES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1987-07-08 EP disclosed
US-4625036-A Antifungal azole compounds IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1986-11-25 US disclosed
EP-0122693-A1 Antifungal di(azolyl)propanol derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1984-10-24 EP disclosed