Bromide

Bromide

SCHEMBL10798602

Br.Br.CCN(CCN1CCC(Sc2nc3ccccc3n2Cc2ccc(F)cc2)CC1)C(=O)O.O

nearest known ligand 0.52

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 11/20 0.52
CYP2D6 P10635 9/20 0.52
LMNA P02545 2/20 0.49
ALDH1A1 P00352 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
TACR2 P21452 1/20 0.46
TACR1 P25103 1/20 0.46
KCNH2 Q12809 6/20 0.46
SSTR5 P35346 2/20 0.46
TP53 P04637 2/20 0.45
CHRM1 P11229 3/20 0.44
NR4A2 P43354 1/20 0.44
MAPT P10636 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9536849 0.82 HRH1 (0.62) HRH1CYP2D6LMNAALDH1A1SMN1; SMN2
SCHEMBL9535641 0.80 SSTR5 (0.52) HRH1CYP2D6LMNAALDH1A1SMN1; SMN2
SCHEMBL9536631 0.75 SSTR5 (0.48) HRH1CYP2D6LMNASMN1; SMN2TACR2
SCHEMBL9537168 0.75 SSTR5 (0.49) HRH1CYP2D6LMNASMN1; SMN2TACR2
SCHEMBL9537373 0.75 TP53 (0.52) HRH1CYP2D6LMNAALDH1A1SMN1; SMN2
SCHEMBL9537130 0.73 KCNH2 (0.63) HRH1CYP2D6LMNAALDH1A1SMN1; SMN2
Hydrochloric Acid SCHEMBL9536691 0.72 CYP2D6 (0.56) HRH1CYP2D6LMNAALDH1A1SMN1; SMN2
SCHEMBL10801027 0.72 TP53 (0.49) HRH1CYP2D6LMNAALDH1A1SMN1; SMN2
SCHEMBL9535858 0.71 PKM (0.51) HRH1CYP2D6LMNAALDH1A1SMN1; SMN2
SCHEMBL1151838 0.70 SSTR5 (0.63) HRH1CYP2D6LMNAALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4695575-A ANTIHISTAMINES JANSSEN PHARMACEUTICA, N.V. (BE) 1987-09-22 US disclosed