SCHEMBL10799296

SCHEMBL10799296

FC(F)(F)c1ccc(-c2nc[nH]n2)nc1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.48
CASP3 P42574 2/20 0.41
KDM4E B2RXH2 2/20 0.40
KIF11 P52732 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
KMT2A Q03164 2/20 0.38
RAB9A P51151 1/20 0.37
ALDH1A1 P00352 2/20 0.36
RECQL P46063 1/20 0.36
TSHR P16473 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
LMNA P02545 1/20 0.35
IDO1 P14902 1/20 0.34
KDM1A O60341 1/20 0.34
MAOB P27338 1/20 0.34
PTGS1 P23219 1/20 0.34
HPGD P15428 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13830687 0.77 NPSR1 (0.50) NPSR1CASP3KDM4EKIF11L3MBTL1
SCHEMBL29595709 0.77 NPSR1 (0.53) NPSR1CASP3KDM4EKIF11L3MBTL1
SCHEMBL811160 0.77 NPSR1 (0.53) NPSR1CASP3KDM4EKIF11L3MBTL1
SCHEMBL2443970 0.77 KIF11 (0.45) KDM4EKIF11RAB9ALMNA
SCHEMBL155254 0.73 METAP2 (0.36) KDM4EALDH1A1LMNA
SCHEMBL27344645 0.71 KIF11 (0.63) NPSR1CASP3KDM4EKIF11KMT2A
SCHEMBL30641506 0.70 NPSR1 (0.45) NPSR1CASP3KDM4EKIF11L3MBTL1
SCHEMBL25405903 0.70 KDM5B (0.36) NPSR1KDM4EL3MBTL1KMT2AALDH1A1
SCHEMBL29690424 0.70 KIF11 (0.61) NPSR1KDM4EKIF11KMT2AIDO1
SCHEMBL28530523 0.70 KIF11 (0.61) NPSR1KDM4EKIF11KMT2AIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0122693-B1 ANTIFUNGAL DI(AZOLYL)PROPANOL DERIVATIVES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1987-07-08 EP disclosed
US-4625036-A Antifungal azole compounds IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1986-11-25 US disclosed
EP-0122693-A1 Antifungal di(azolyl)propanol derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1984-10-24 EP disclosed