SCHEMBL10812902

SCHEMBL10812902

CC(=O)CC(=O)c1ccc(C)nc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.58
HDAC6 Q9UBN7 1/20 0.58
KDM4E B2RXH2 2/20 0.51
MAPT P10636 3/20 0.42
ALDH1A1 P00352 3/20 0.42
KMT2A Q03164 3/20 0.41
KCNQ3 O43525 1/20 0.41
KCNQ2 O43526 1/20 0.41
NPC1 O15118 2/20 0.41
CYP19A1 P11511 1/20 0.41
PRKAB2 O43741 1/20 0.40
PRKAG1 P54619 1/20 0.40
PRKAA2 P54646 1/20 0.40
PRKAA1 Q13131 1/20 0.40
PRKAG3 Q9UGI9 1/20 0.40
PRKAG2 Q9UGJ0 1/20 0.40
PRKAB1 Q9Y478 1/20 0.40
POLB P06746 1/20 0.40
LMNA P02545 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15136337 0.83 HDAC1 (0.55) HDAC1HDAC6KDM4EMAPTALDH1A1
SCHEMBL11620450 0.82 HDAC1 (0.50) HDAC1HDAC6KDM4EMAPTALDH1A1
SCHEMBL4734775 0.82 HDAC1 (0.54) HDAC1HDAC6KDM4EMAPTALDH1A1
Hydrochloric Acid SCHEMBL9672401 0.81 HDAC1 (0.53) HDAC1HDAC6KDM4EMAPTALDH1A1
Hydrochloric Acid SCHEMBL3231047 0.81 HDAC1 (0.53) HDAC1HDAC6KDM4EMAPTALDH1A1
SCHEMBL2632670 0.81 HDAC1 (0.56) HDAC1HDAC6KDM4EMAPTALDH1A1
SCHEMBL3464701 0.80 NAPRT (0.56) MAPTALDH1A1KMT2AKCNQ3KCNQ2
SCHEMBL29939457 0.80 HDAC1 (0.51) HDAC1HDAC6KDM4EMAPTALDH1A1
SCHEMBL10662120 0.80 HDAC1 (0.51) HDAC1HDAC6KDM4EMAPTALDH1A1
SCHEMBL4745823 0.80 PLOD2 (0.60) HDAC1HDAC6KDM4EMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4650806-A Cardiotonic 5-(heterylcarbonyl)-pyridones STERLING DRUG INC. (US) 1987-03-17 US disclosed
EP-0191298-A2 1,6 -Naphthyridin-2(1H) - ones useful as cardiotonics and preparation thereof STERLING DRUG INC. (US) 1986-08-20 EP disclosed
US-4567186-A 5-Heteryl-1,6-naphthyridin-2(1H)-ones, cardiotonic use thereof and intermediates therefor STERLING DRUG INC. (US) 1986-01-28 US disclosed
US-4088764-A CARDIOVASCULAR DISORDERS, BETA-ADRENERGIC BLOCKING AGENTS, ANTIARRHYTHMIC AGENTS CASSELLA FARBWERKE MAINKUR AKTIENGESELLSCHAFT (DT) 1978-05-09 US disclosed
US-4066768-A ADRENERGIC BLOCKING AGENTS, ANTIARRHYTHMIC CASSELLA FARBWERKE MAINKUR AKTIENGESELLSCHAFT (DT) 1978-01-03 US disclosed
US-3969363-A CARDIOVASCULAR DISORDERS CASSELLA FARBWERKE MAINKUR AKTIENGESELLSCHAFT (DT) 1976-07-13 US disclosed