SCHEMBL10813693

SCHEMBL10813693

COc1cc([N+](=O)[O-])c(Nc2ccccc2)cn1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 1/20 0.52
L3MBTL1 Q9Y468 5/20 0.51
ALDH1A1 P00352 4/20 0.51
TDP1 Q9NUW8 3/20 0.51
MAPK1 P28482 2/20 0.51
CASP7 P55210 1/20 0.51
MAPT P10636 7/20 0.49
HPGD P15428 2/20 0.49
POLB P06746 1/20 0.48
AKR1C3 P42330 2/20 0.46
AKR1C2 P52895 2/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
AKR1B10 O60218 1/20 0.46
AKR1B1 P15121 1/20 0.46
AKR1C4 P17516 1/20 0.46
AKR1C1 Q04828 1/20 0.46
GAA P10253 2/20 0.46
LMNA P02545 1/20 0.46
HTT P42858 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10635085 0.80 AKR1C3 (0.54) ALDH1A1TDP1MAPK1MAPTHPGD
SCHEMBL10635096 0.78 ERN1 (0.47) L3MBTL1ALDH1A1TDP1MAPK1MAPT
SCHEMBL7990043 0.77 ALDH1A1 (0.57) HCAR3L3MBTL1ALDH1A1TDP1MAPK1
SCHEMBL30615538 0.76 ABCG2 (0.49) L3MBTL1ALDH1A1TDP1MAPK1CASP7
SCHEMBL21463999 0.76 ABCG2 (0.49) L3MBTL1ALDH1A1TDP1MAPK1CASP7
SCHEMBL3996405 0.76 ALDH1A1 (0.58) HCAR3L3MBTL1ALDH1A1TDP1MAPK1
SCHEMBL6179431 0.76 AKR1C3 (0.74) HCAR3L3MBTL1ALDH1A1TDP1MAPK1
SCHEMBL4944345 0.76 L3MBTL1 (0.60) L3MBTL1ALDH1A1TDP1MAPK1CASP7
SCHEMBL9943157 0.74 L3MBTL1 (0.70) HCAR3L3MBTL1ALDH1A1TDP1MAPK1
SCHEMBL7976555 0.74 TDP1 (0.54) HCAR3L3MBTL1ALDH1A1TDP1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4698430-A ANTIDEPRESSANT A. H. ROBINS COMPANY, INC. (US) 1987-10-06 US disclosed
US-4558132-A ANTIDEPRESSANTS A. H. ROBINS COMPANY, INCORPORATED (US) 1985-12-10 US disclosed
EP-0099614-A2 Nitro, amino and aroylamino-N-phenylpyridinamines and their use in a process for preparing pyrido(1,4)benzodiazapines A.H. ROBINS COMPANY, INCORPORATED (US) 1984-02-01 EP disclosed