SCHEMBL10822154

SCHEMBL10822154

O=[C]C(c1nnn[nH]1)N(Cc1ccccc1)C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
LMNA P02545 4/20 0.37
ALDH1A1 P00352 2/20 0.37
KDM4E B2RXH2 1/20 0.37
ATM Q13315 1/20 0.36
HCAR3 P49019 1/20 0.35
POLB P06746 1/20 0.35
HSD17B10 Q99714 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
CA12 O43570 1/20 0.33
CA9 Q16790 1/20 0.33
HPGD P15428 1/20 0.32
FNTA P49354 1/20 0.32
FNTB P49356 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22370925 0.81 MEN1 (0.48) MEN1KMT2ALMNAALDH1A1ATM
SCHEMBL14910876 0.76 MEN1 (0.43) MEN1KMT2ALMNAALDH1A1ATM
SCHEMBL531534 0.69 MEN1 (0.37) MEN1KMT2ALMNAALDH1A1ATM
SCHEMBL19354535 0.66 IDO1 (0.43) KDM4EL3MBTL1
SCHEMBL19354261 0.66 IDO1 (0.43) KDM4EL3MBTL1
SCHEMBL11326774 0.66 ALDH1A1 (0.38) KMT2AALDH1A1KDM4EATMPOLB
SCHEMBL11528941 0.66 CYP1A2 (0.42)
SCHEMBL2093344 0.65 CYP1A2 (0.39)
SCHEMBL11568927 0.65 TDP1 (0.55) MEN1KMT2ALMNAALDH1A1ATM
SCHEMBL5908164 0.65 CYP1A2 (0.45) ALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4604386-A CONTROL OF GRAMPOSITIVE BACTERIA ELI LILLY AND COMPANY (US) 1986-08-05 US disclosed
EP-0168222-A2 3-(Alkynylalkyloxy) Cephalosporins ELI LILLY AND COMPANY (US) 1986-01-15 EP disclosed