SCHEMBL10829068

SCHEMBL10829068

Nc1nc(O)c2cc(CN(CCF)c3ccc(C(=O)N[C@H](CCC(=O)O)C(=O)O)cc3)ccc2n1

nearest known ligand 0.67

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
DHFR P00374 7/20 0.64
TYMS P04818 4/20 0.57
ATIC P31939 2/20 0.55
GART P22102 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10828707 1.00 DHFR (0.64) DHFRTYMSATICGART
SCHEMBL10829048 0.91 DHFR (0.60) DHFRTYMS
SCHEMBL10828960 0.89 DHFR (0.78) DHFRTYMSATIC
SCHEMBL6579718 0.88 DHFR (0.78) DHFRTYMS
SCHEMBL10828939 0.87 DHFR (0.60) DHFRTYMSATICGART
SCHEMBL6337570 0.86 DHFR (0.77) DHFRTYMSATICGART
SCHEMBL10828697 0.86 DHFR (0.53) DHFRTYMS
SCHEMBL10828701 0.86 DHFR (0.53) DHFRTYMS
SCHEMBL10829007 0.83 ATIC (0.57) DHFRTYMSATICGART
SCHEMBL24629149 0.82 DHFR (0.70) DHFRTYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4564616-A Anti-cancer quinazoline derivatives NATIONAL RESEARCH DEVELOPMENT CORPORATION (GB) 1986-01-14 US disclosed
EP-0031237-B1 QUINAZOLINE DERIVATIVES, PROCESSES FOR THEIR PREPARATION, COMPOSITIONS CONTAINING THEM AND THEIR USE AS ANTI-CANCER AGENTS NATIONAL RESEARCH DEVELOPMENT CORPORATION (GB) 1984-10-17 EP disclosed
US-4447608-A ANTITUMOR AGENTS NATIONAL RESEARCH DEVELOPMENT CORPORATION (GB) 1984-05-08 US disclosed
EP-0031237-A1 Quinazoline derivatives, processes for their preparation, compositions containing them and their use as anti-cancer agents NATIONAL RESEARCH DEVELOPMENT CORPORATION (GB) 1981-07-01 EP disclosed