SCHEMBL10832811

SCHEMBL10832811

COc1c(OC)c(OC(C)=O)c2c(Sc3c(Cl)cccc3Cl)cccc2c1OC(C)=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB11 O95342 1/20 0.46
ALDH1A1 P00352 3/20 0.36
USP7 Q93009 3/20 0.36
NLRP3 Q96P20 1/20 0.35
MAPT P10636 4/20 0.34
HTT P42858 3/20 0.34
POLB P06746 2/20 0.34
TSHR P16473 1/20 0.34
USP47 Q96K76 1/20 0.34
KDM4E B2RXH2 5/20 0.33
TUBB4A P04350 2/20 0.33
TUBB P07437 2/20 0.33
TUBA3C P0DPH7 2/20 0.33
TUBA1B P68363 2/20 0.33
TUBA4A P68366 2/20 0.33
TUBB4B P68371 2/20 0.33
TUBB3 Q13509 2/20 0.33
TUBB2A Q13885 2/20 0.33
TUBB8 Q3ZCM7 2/20 0.33
TUBA3E Q6PEY2 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9642267 0.84 ABCB11 (0.55) ABCB11ALDH1A1NLRP3MAPTHTT
SCHEMBL9713640 0.83 ALDH1A1 (0.38) ABCB11ALDH1A1MAPTHTTPOLB
SCHEMBL9644096 0.82 ABCB11 (0.42) ABCB11ALDH1A1MAPTHTTKDM4E
SCHEMBL10832739 0.82 ABCB11 (0.52) ABCB11USP7MAPTTUBB4ATUBB
SCHEMBL10833190 0.80 ABCB11 (0.40) ABCB11ALDH1A1NLRP3MAPTHTT
SCHEMBL10832729 0.79 ABCB11 (0.39) ABCB11ALDH1A1MAPTPOLBKDM4E
SCHEMBL9643904 0.78 ABCB11 (0.51) ABCB11NLRP3MAPTHTTPOLB
SCHEMBL10892237 0.76 KDM4E (0.41) ABCB11ALDH1A1MAPTHTTPOLB
SCHEMBL9643403 0.75 ABCB11 (0.48) ABCB11ALDH1A1NLRP3MAPTHTT
SCHEMBL9641706 0.74 ABCB11 (0.53) ABCB11ALDH1A1MAPTHTTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4593120-A Naphthalene-1,4-dicarboxylic acid group SYNTEX (U.S.A.) INC. (US) 1986-06-03 US disclosed
EP-0107512-B1 1,4-ACYLOXYNAPHTHALENE DERIVATIVES, TOPICAL COMPOSITIONS CONTAINING THEM, METHODS FOR THEIR PREPARATION, AND INTERMEDIATES THEREFOR SYNTEX (U.S.A.) INC. (US) 1986-02-26 EP disclosed
US-4466981-A Naphthalene anti-psoriatic agents SYNTEX (U.S.A.) INC. (US) 1984-08-21 US disclosed
EP-0107512-A1 1,4-Acyloxynaphthalene derivatives, topical compositions containing them, methods for their preparation, and intermediates therefor SYNTEX (U.S.A.) INC. (US) 1984-05-02 EP disclosed