SCHEMBL10836637

SCHEMBL10836637

COc1ccc2c(c1Br)CCC(C#N)C2C#N

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 2/20 0.35
CYP1A2 P05177 1/20 0.34
CYP19A1 P11511 2/20 0.32
AR P10275 2/20 0.32
DRD2 P14416 3/20 0.32
DRD3 P35462 3/20 0.32
HSD11B1 P28845 1/20 0.31
DRD4 P21917 2/20 0.31
STS P08842 1/20 0.31
KDM4E B2RXH2 1/20 0.31
HTR2A P28223 1/20 0.30
MTNR1A P48039 1/20 0.30
MTNR1B P49286 1/20 0.30
CHRM2 P08172 1/20 0.30
CHRM1 P11229 1/20 0.30
CHRM3 P20309 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10504881 0.84 PARP1 (0.42) ADRA1ADRD2DRD3KDM4E
SCHEMBL10836323 0.83 CYP19A1 (0.46) ADRA1ACYP1A2CYP19A1DRD2DRD3
SCHEMBL9457736 0.78 CYP1A2 (0.42) ADRA1ACYP1A2CYP19A1ARDRD2
SCHEMBL10835925 0.77 ADRA1A (0.43) ADRA1ACYP1A2CYP19A1ARDRD2
SCHEMBL29944713 0.73 POLL (0.48) ADRA1ACYP1A2CYP19A1DRD2DRD3
SCHEMBL20269738 0.73 POLL (0.48) ADRA1ACYP1A2CYP19A1DRD2DRD3
SCHEMBL10504886 0.71 CA1 (0.43) DRD2MTNR1AMTNR1B
SCHEMBL9458168 0.69 DRD2 (0.44) DRD2DRD3CHRM2CHRM1CHRM3
SCHEMBL10836107 0.69 CYP19A1 (0.46) CYP19A1DRD2DRD3
SCHEMBL9361544 0.68 CA1 (0.45) ADRA1ACYP1A2CYP19A1DRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4618683-A Tetrahydro-6,7-dimethoxy-1H-benz[e]isoinodolines useful in the treatment of hypertension and as sedatives ABBOTT LABORATORIES (US) 1986-10-21 US disclosed