SCHEMBL10837643

SCHEMBL10837643

O=C1c2ccccc2C(=O)N1CCNc1ccsc1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RPS6KA2 Q15349 3/20 0.44
GLS O94925 1/20 0.44
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
POLB P06746 2/20 0.43
CASP1 P29466 1/20 0.43
OGA O60502 1/20 0.42
HEXA P06865 1/20 0.42
HEXB P07686 1/20 0.42
MAPT P10636 2/20 0.42
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
HTT P42858 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
ACHE P22303 4/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16087635 0.80 RPS6KA2 (0.56) RPS6KA2GLSMEN1KMT2AMAPT
SCHEMBL3062593 0.76 RPS6KA2 (0.73) RPS6KA2KMT2APOLBALDH1A1HPGD
SCHEMBL8436723 0.73 CASP3 (0.57) GLSMEN1KMT2APOLBCASP1
SCHEMBL805142 0.73 OGA (0.70) GLSOGAHEXAHEXBSMN1; SMN2
SCHEMBL2754749 0.72 RAB9A (0.55) RPS6KA2GLSMEN1KMT2APOLB
SCHEMBL11237861 0.72 CYP1A2 (0.57) RPS6KA2MEN1KMT2AMAPTALDH1A1
SCHEMBL10819269 0.72 RPS6KA2 (0.74) RPS6KA2MEN1KMT2APOLBHEXA
SCHEMBL28776422 0.71 CES1 (0.60) RPS6KA2MEN1KMT2APOLBHEXA
SCHEMBL7973833 0.71 OGA (0.68) GLSOGAHEXAHEXBSMN1; SMN2
SCHEMBL6699936 0.70 GLS (0.71) GLSMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4608383-A Cardioactive pyrazole and imidazole aryloxypropanolamines BOEHRINGER MANNHEIM GMBH (DE) 1986-08-26 US disclosed
US-4438128-A ADRENERGIC BLOCKERS BOEHRINGER MANNHEIM GMBH (DE) 1984-03-20 US disclosed