SCHEMBL10838457

SCHEMBL10838457

NC(=O)c1ccc(Nc2ccc3ccccc3n2)cc1

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 1/20 0.55
NPC1 O15118 7/20 0.51
RAB9A P51151 6/20 0.51
KMT2A Q03164 1/20 0.50
RHOA P61586 1/20 0.49
AURKA O14965 2/20 0.48
AURKB Q96GD4 1/20 0.47
MAPT P10636 2/20 0.47
KDM4E B2RXH2 1/20 0.47
NCF1 P14598 1/20 0.46
MAPK8 P45983 1/20 0.46
MAPK10 P53779 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
SIRT2 Q8IXJ6 1/20 0.45
SIRT1 Q96EB6 1/20 0.45
SIRT3 Q9NTG7 1/20 0.45
KDM1A O60341 1/20 0.44
MKNK1 Q9BUB5 1/20 0.44
MKNK2 Q9HBH9 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4494871 0.79 KMT2A (0.58) NPC1RAB9AKMT2ARHOAAURKA
SCHEMBL4812645 0.79 NCF1 (0.53) NPC1RAB9AKMT2ARHOAMAPT
SCHEMBL27960243 0.78 RHOA (0.55) NPC1RAB9AKMT2ARHOAAURKA
SCHEMBL29833517 0.78 NCF1 (0.61) ROCK1NPC1RAB9AKMT2ARHOA
SCHEMBL396525 0.78 NCF1 (0.61) ROCK1NPC1RAB9AKMT2ARHOA
SCHEMBL11566043 0.77 GRM5 (0.60) NPC1RAB9AKMT2AMAPTKDM4E
SCHEMBL30534868 0.77 DNMT1 (0.59) NPC1RAB9AKMT2AMAPTKDM4E
SCHEMBL21446750 0.77 RAB9A (0.73) NPC1RAB9AKMT2AMAPTKDM4E
SCHEMBL9965273 0.76 NPC1 (0.64) ROCK1NPC1RAB9AKMT2AKDM4E
SCHEMBL29110577 0.76 NPC1 (0.58) NPC1RAB9AKMT2ARHOAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4610991-A Antihypertensive pyridylaminobenzamide compounds STERLING DRUG INC. (US) 1986-09-09 US disclosed
EP-0098951-A2 Aminobenzamide derivatives and preparation thereof STERLING DRUG INC. (US) 1984-01-25 EP disclosed