SCHEMBL10842020

SCHEMBL10842020

CC(C)(C)OC(=O)O/N=C(/C(N)=O)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.50
GAA P10253 1/20 0.50
ELANE P08246 1/20 0.41
TNF P01375 1/20 0.41
KLF5 Q13887 1/20 0.41
NOD1 Q9Y239 1/20 0.41
USP2 O75604 1/20 0.41
ALDH1A1 P00352 3/20 0.40
TSHR P16473 2/20 0.40
HSD17B10 Q99714 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
HPGD P15428 1/20 0.38
AAK1 Q2M2I8 1/20 0.37
MAPT P10636 2/20 0.37
POLB P06746 1/20 0.37
CYP3A4 P08684 1/20 0.37
PARP1 P09874 1/20 0.37
RECQL P46063 1/20 0.37
BLM P54132 1/20 0.37
PMP22 Q01453 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10842026 1.00 CYP2C19 (0.50) CYP2C19GAAELANETNFKLF5
SCHEMBL10173004 0.84 TNF (0.57) GAATNFKLF5NOD1USP2
SCHEMBL11321880 0.82 AAK1 (0.46) ELANETNFKLF5NOD1USP2
SCHEMBL25314654 0.78 CYP2C19 (0.58) CYP2C19GAAELANETNFKLF5
SCHEMBL11521468 0.78 CYP2C19 (0.58) CYP2C19GAAELANETNFKLF5
SCHEMBL11324498 0.77 CES2 (0.46) CYP2C19ELANETNFKLF5NOD1
SCHEMBL11324501 0.77 CES2 (0.46) CYP2C19ELANETNFKLF5NOD1
SCHEMBL7045591 0.77 ELANE (0.41) CYP2C19ELANETNFKLF5NOD1
SCHEMBL7130236 0.76 CYP2C19 (0.60) CYP2C19GAATNFKLF5NOD1
SCHEMBL22758099 0.76 CYP2C19 (0.60) CYP2C19GAATNFKLF5NOD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4593098-A Piperazinone and piperazine polypeptides THE UPJOHN COMPANY (US) 1986-06-03 US disclosed
US-4534897-A Piperazinone, piperazine, 1,4-diazepin-2-one and 1,4-diazepine intermediate compounds THE UPJOHN COMPANY (US) 1985-08-13 US disclosed
US-4251438-A ANALGESICS, PSYCHOTHERAPEUTIC AGENTS THE UPJOHN COMPANY (US) 1981-02-17 US disclosed