SCHEMBL10847722

SCHEMBL10847722

CCOC(=O)C1=C(C)NC(C)=C(C(=O)OCCN2CCC(C(c3ccccc3)c3ccccc3)CC2)C1c1cccc(Cl)c1Cl

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.59
CYP3A4 P08684 3/20 0.59
ABCB11 O95342 3/20 0.59
TBXA2R P21731 3/20 0.59
ADRA1A P35348 3/20 0.59
SLC6A3 Q01959 3/20 0.59
KDM4E B2RXH2 2/20 0.59
MEN1 O00255 2/20 0.59
CYP1A2 P05177 2/20 0.59
CYP2C19 P33261 2/20 0.59
KMT2A Q03164 2/20 0.59
HIF1A Q16665 2/20 0.59
HSD17B10 Q99714 2/20 0.59
LMNA P02545 2/20 0.59
TSHR P16473 2/20 0.59
ABCB1 P08183 2/20 0.59
ADORA3 P0DMS8 2/20 0.59
ADRB3 P13945 2/20 0.59
OPRK1 P41145 2/20 0.59
SCN5A Q14524 2/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10367174 0.89 CYP2C9 (0.60) CYP2C9CYP3A4ABCB11TBXA2RADRA1A
SCHEMBL10366636 0.83 CYP2C9 (0.59) CYP2C9CYP3A4ABCB11TBXA2RADRA1A
SCHEMBL10367481 0.83 ADRA1A (0.61) CYP2C9CYP3A4ABCB11TBXA2RADRA1A
SCHEMBL10365985 0.82 SLC6A3 (0.50) CYP2C9CYP3A4ABCB11TBXA2RADRA1A
SCHEMBL10930978 0.82 CYP2C9 (0.57) CYP2C9CYP3A4ABCB11TBXA2RADRA1A
Hydrochloric Acid SCHEMBL10928623 0.81 CYP2C9 (0.56) CYP2C9CYP3A4ABCB11TBXA2RADRA1A
SCHEMBL7279434 0.79 ABCB11 (0.54) CYP2C9CYP3A4ABCB11TBXA2RADRA1A
SCHEMBL10741475 0.79 ADRA1A (0.63) CYP2C9CYP3A4ABCB11TBXA2RADRA1A
SCHEMBL29756037 0.79 KDM4E (0.90) CYP2C9CYP3A4ABCB11TBXA2RADRA1A
SCHEMBL3029888 0.79 KDM4E (0.90) CYP2C9CYP3A4ABCB11TBXA2RADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4603135-A HYPOTENSIVE AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1986-07-29 US disclosed